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Found 332 of affinity data for UniProtKB/TrEMBL: P06536
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86689(CAS_84371-65-3 | NSC_55245 | RU-486)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86690(A 348441 | A-348441)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50499243(CHEMBL3735203)
Affinity DataKi:  8.5nMAssay Description:Antagonist activity at glucocorticoid receptor in rat H4IIEC3 cells assessed as glucocorticoid-induced TAT activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50265673(CHEMBL4068611)
Affinity DataKi:  12nMAssay Description:Antagonist activity at rat glucocorticoid receptor in primary hepatocytes assessed as dexamethasone-induced tyrosine amino transferase activity prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50265674(CHEMBL3734774)
Affinity DataKi:  13nMAssay Description:Antagonist activity at glucocorticoid receptor in rat primary hepatocytes assessed as inhibition of glucocorticoid-induced TAT activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50499243(CHEMBL3735203)
Affinity DataKi:  150nMAssay Description:Antagonist activity at glucocorticoid receptor in rat primary hepatocytes assessed as inhibition of glucocorticoid-induced TAT activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597074(CHEMBL5197264)
Affinity DataKi:  1.96E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597080(CHEMBL5207249)
Affinity DataKi:  2.22E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597079(CHEMBL5207123)
Affinity DataKi:  2.54E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597071(CHEMBL5191961)
Affinity DataKi:  2.90E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597078(CHEMBL5181002)
Affinity DataKi:  2.91E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597070(CHEMBL5186524)
Affinity DataKi:  3.79E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597068(CHEMBL5201004)
Affinity DataKi:  4.00E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597081(CHEMBL5184647)
Affinity DataKi:  4.15E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597087(CHEMBL5181278)
Affinity DataKi:  4.32E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597077(CHEMBL5172350)
Affinity DataKi:  4.50E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597076(CHEMBL5176336)
Affinity DataKi:  4.72E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597083(CHEMBL5171957)
Affinity DataKi:  5.52E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50004519(CHEMBL2181929)
Affinity DataKi:  8.42E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597082(CHEMBL5204612)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597075(CHEMBL5186231)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597073(CHEMBL5182687)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597072(CHEMBL5173089)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597067(CHEMBL5182675)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597069(CHEMBL5208644)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597085(CHEMBL5183454)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597086(CHEMBL5187656)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50597084(CHEMBL5174401)
Affinity DataKi:  1.36E+5nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM141379(US8916600, 13 | US9738632, Example 13)
Affinity DataIC50:  0.100nMAssay Description:Transrepression of glucocorticoid receptor in Wistar rat PBMC assessed as inhibition of LPS induced TNF alpha release preincubated for 45 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50354849(CCI-18781 | Cutivate | FLUTICASONE PROPIONATE | Fl...)
Affinity DataIC50:  0.140nMAssay Description:Transrepression of glucocorticoid receptor in Wistar rat PBMC assessed as inhibition of LPS induced TNF alpha release preincubated for 45 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50250112(CHEMBL4072756)
Affinity DataIC50:  0.140nMAssay Description:Transrepression of glucocorticoid receptor in Wistar rat PBMC assessed as inhibition of LPS induced TNF alpha release preincubated for 45 mins follow...More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50577704(CHEMBL4863316)
Affinity DataIC50:  0.158nMAssay Description:Agonist activity at glucocorticoid receptor in rat INS-1 832/13 cells transfected with CCL2-promoter luciferase plasmid construct assessed as reducti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50577694(CHEMBL4877227)
Affinity DataIC50:  0.200nMAssay Description:Agonist activity at glucocorticoid receptor in rat INS-1 832/13 cells transfected with CCL2-promoter luciferase plasmid construct assessed as reducti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM19235(2-{5-[4-({[(2,4-difluorophenyl)methyl](3-methanesu...)
Affinity DataIC50:  0.200nMpH: 8.0 T: 2°CAssay Description:For compounds able to displace the radiolabeled ligand (competitor) from the receptor an IC50 value (the concentration required to inhibit 50% of the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM19205((1R)-1-[(4aR,5S)-1-(4-fluorophenyl)-4a-methyl-1H,4...)
Affinity DataIC50:  0.251nMAssay Description:Agonist activity at glucocorticoid receptor in rat INS-1 832/13 cells transfected with CCL2-promoter luciferase plasmid construct assessed as reducti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM141378(US8916600, 12 | US9738632, Example 12)
Affinity DataIC50:  0.290nMAssay Description:Transrepression of glucocorticoid receptor in Wistar rat PBMC assessed as inhibition of LPS induced TNF alpha release preincubated for 45 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM141372(US8916600, 6 | US9738632, Example 6)
Affinity DataIC50:  0.300nMAssay Description:Transrepression of glucocorticoid receptor in Wistar rat PBMC assessed as inhibition of LPS induced TNF alpha release preincubated for 45 mins follow...More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50594611(CHEMBL5196090)
Affinity DataIC50:  0.316nMAssay Description:Agonist activity at glucocorticoid receptor in rat INS-1 832/13 cells transfected with CCL2-promoter luciferase plasmid construct assessed as reducti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM141368(US8916600, 2 | US8916600, 3 | US9738632, Example 2)
Affinity DataIC50:  0.340nMAssay Description:Transrepression of glucocorticoid receptor in Wistar rat PBMC assessed as inhibition of LPS induced TNF alpha release preincubated for 45 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50250124(CHEMBL4099639)
Affinity DataIC50:  0.560nMAssay Description:Transrepression of glucocorticoid receptor in Wistar rat PBMC assessed as inhibition of LPS induced TNF alpha release preincubated for 45 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50594601(CHEMBL5181366)
Affinity DataIC50:  0.631nMAssay Description:Agonist activity at glucocorticoid receptor in rat INS-1 832/13 cells transfected with CCL2-promoter luciferase plasmid construct assessed as reducti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50153502(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50014432(CHEMBL3261407)
Affinity DataIC50:  0.900nMAssay Description:Agonist activity at glucocorticoid receptor in rat PBMC assessed as inhibition of LPS-stimulated TNF-alpha releaseMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM19234(4-{4-[3-(4-{[benzyl(3-methanesulfonamido-2-methylp...)
Affinity DataIC50:  1nMpH: 8.0 T: 2°CAssay Description:For compounds able to displace the radiolabeled ligand (competitor) from the receptor an IC50 value (the concentration required to inhibit 50% of the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50:  1.30nMAssay Description:Agonist activity at glucocorticoid receptor in rat INS-1 832/13 cells transfected with CCL2-promoter luciferase plasmid construct assessed as reducti...More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  1.40nMpH: 8.0 T: 2°CAssay Description:For compounds able to displace the radiolabeled ligand (competitor) from the receptor an IC50 value (the concentration required to inhibit 50% of the...More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50054959((4aS,4bR,5S,6aS,6bR,9aR)-4b-Fluoro-5-hydroxy-4a,6a...)
Affinity DataIC50:  1.60nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50054966((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-4a...)
Affinity DataIC50:  1.70nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50407988(CHEMBL2112857)
Affinity DataIC50:  1.80nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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