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TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM697956(1 alpha, 25 (OH)2 VD2 | US20240317663, Compound Ia)
Affinity DataEC50:  10.8nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
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TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM697957(19-nor-1 alpha, 25 (OH)2 VD3 | US20240317663, Comp...)
Affinity DataEC50:  4.80nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50619813(US20240317663, Compound IIa | CHEMBL5408377)
Affinity DataEC50:  7.5nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
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TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50619817(US20240317663, Compound IIIa | CHEMBL5434792)
Affinity DataEC50:  7.40nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50619814(US20240317663, Compound IIb | CHEMBL5423207)
Affinity DataEC50:  17.4nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50619818(US20240317663, Compound IIIb | CHEMBL5404109)
Affinity DataEC50:  6.70nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50619815(US20240317663, Compound epi-IIb | CHEMBL5395581)
Affinity DataEC50:  518nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM697963(des-D-19-nor-bC | US20240317663, Compound IV | BDB...)
Affinity DataEC50:  84nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
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TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM697964(des-D-19-nor-aB | US20240317663, Compound V)
Affinity DataEC50:  243nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM697963(des-D-19-nor-bC | US20240317663, Compound IV | BDB...)
Affinity DataEC50:  50.3nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM697966(des-D-19-nor-cA | US20240317663, Compound VII)
Affinity DataEC50: >5.00E+3nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM697967(des-D-19-nor-OH c | US20240317663, Compound VIII)
Affinity DataEC50: >5.00E+3nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM697968(des-D-19-nor-CbB | US20240317663, Compound IX)
Affinity DataEC50:  922nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50619822(US20240317663, Compound epi-IX | CHEMBL5405063)
Affinity DataEC50:  846nMAssay Description:A VDR ligand binding domain tagged with GST (VDR-LBD(GST)), a fluorescein-TRAP220/DRIP-2-bound coactivator peptide (Fluorescein-peptide), LanthaScree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50242220(CHEMBL4066573)
Affinity DataKd:  142nMAssay Description:Binding affinity to recombinant human GST-tagged VDR LBD (156 to 453 residues) expressed in Echerichia coli BL21 star (DE3) after 40 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50242218(CHEMBL4086339)
Affinity DataKd:  197nMAssay Description:Binding affinity to recombinant human GST-tagged VDR LBD (156 to 453 residues) expressed in Echerichia coli BL21 star (DE3) after 40 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50242219(CHEMBL4067602)
Affinity DataKd: >2.00E+3nMAssay Description:Binding affinity to recombinant human GST-tagged VDR LBD (156 to 453 residues) expressed in Echerichia coli BL21 star (DE3) after 40 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50254160(CHEMBL4062601)
Affinity DataEC50:  4.10E+3nMAssay Description:Agonist activity at vitamin D receptor (unknown origin) expressed in HEK293 cells co-expressing pCMX-RXRalpha and pCMX-beta-galactosidase assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50254164(CHEMBL4075325)
Affinity DataEC50:  3.70E+3nMAssay Description:Agonist activity at vitamin D receptor (unknown origin) expressed in HEK293 cells co-expressing pCMX-RXRalpha and pCMX-beta-galactosidase assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50254165(CHEMBL4080769)
Affinity DataEC50:  850nMAssay Description:Agonist activity at vitamin D receptor (unknown origin) expressed in HEK293 cells co-expressing pCMX-RXRalpha and pCMX-beta-galactosidase assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256289(CHEMBL4072930)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256290(CHEMBL4093629)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256291(CHEMBL4096970)
Affinity DataEC50:  6.03E+3nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256292(CHEMBL4086285)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256293(CHEMBL4075991)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256294(CHEMBL4073404)
Affinity DataEC50:  1.63E+3nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256295(CHEMBL4101788)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256296(CHEMBL4063772)
Affinity DataEC50:  21nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256297(CHEMBL4091572)
Affinity DataEC50:  860nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256308(CHEMBL4101251)
Affinity DataEC50:  66nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256309(CHEMBL4074522)
Affinity DataEC50:  450nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256310(CHEMBL4063153)
Affinity DataEC50:  53nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256333(CHEMBL4085761)
Affinity DataEC50:  96nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256307(CHEMBL4097419)
Affinity DataEC50:  89nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256334(CHEMBL4075907)
Affinity DataEC50:  11nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256339(CHEMBL4074357)
Affinity DataEC50:  5nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256336(CHEMBL4102275)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256337(CHEMBL4078012)
Affinity DataEC50:  1.08E+3nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256340(CHEMBL4101362)
Affinity DataEC50:  238nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256341(CHEMBL4085890)
Affinity DataEC50:  82nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256342(CHEMBL4083376)
Affinity DataEC50:  156nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256343(CHEMBL4078953)
Affinity DataEC50:  2.65E+3nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256344(CHEMBL4094053)
Affinity DataEC50:  5.90E+3nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256345(CHEMBL4083785)
Affinity DataEC50:  520nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256346(CHEMBL4079382)
Affinity DataEC50:  26nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256347(CHEMBL4084799)
Affinity DataEC50:  2.49E+3nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50256338(CHEMBL4103687)
Affinity DataEC50:  8.5nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50281390(CHEMBL4159525)
Affinity DataEC50:  0.140nMAssay Description:Transactivation of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-RXRalpha and MH100(UAS) X 4tk-LUC reporter plasmid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Kanagawa University

US Patent
LigandPNGBDBM50281390(CHEMBL4159525)
Affinity DataEC50: >1.20nMAssay Description:Transactivation of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-SRC-1 and MH100(UAS) X 4tk-LUC reporter plasmid ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2020
Entry Details Article
PubMed
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