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TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50599148BDBM50599148(CHEMBL5188777)
Affinity DataKd:  0.00500nMAssay Description:Displacement of ARC-1063 fluorescent probe from recombinant human PKAC-alpha assessed as dissociation equilibrium constant preincubated for 1 hr foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50599153BDBM50599153(CHEMBL5196521)
Affinity DataKi:  0.00700nMAssay Description:Covalent inhibition of human recombinant PKAC-alpha assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50599147BDBM50599147(CHEMBL5201435)
Affinity DataKd:  0.0190nMAssay Description:Displacement of ARC-1063 fluorescent probe from recombinant human PKAC-alpha assessed as dissociation equilibrium constant preincubated for 1 hr foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50599152BDBM50599152(CHEMBL5179794)
Affinity DataKi:  0.0230nMAssay Description:Covalent inhibition of human recombinant PKAC-alpha assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587772BDBM50587772(CHEMBL5185265)
Affinity DataKd:  0.0420nMAssay Description:Displacement of mAb(D38C6)-BTN from human recombinant PKAc alpha incubated for 15 mins by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 258601BDBM258601(US9493490, Example 13 | US9493490, 6-(4-(aminometh...)
Affinity DataIC50: 0.0550nMT: 2°CAssay Description:Phosphorylation of activity of ROCK1 and ROCK2 and those of other kinases, AKT1, GRK2, PKA, PKCa and RSK1 were performed by Reaction Biology (Malvern...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50188913BDBM50188913(N-((S)-1-amino-3-(2,4-dichlorophenyl)propan-2-yl)-...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50599149BDBM50599149(CHEMBL5174535)
Affinity DataKi:  0.630nMAssay Description:Covalent inhibition of human recombinant PKAC-alpha assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50599146BDBM50599146(CHEMBL5189362)
Affinity DataKd:  0.630nMAssay Description:Displacement of ARC-1063 fluorescent probe from recombinant human PKAC-alpha assessed as dissociation equilibrium constant preincubated for 1 hr foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 139540BDBM139540(US8889696, Staurosporine | US9051313, Staurosporin...)
Affinity DataIC50: 0.678nMAssay Description:Compounds as a powder were dissolved in dimethyl sulfoxide to make a 10 mM stock. Compounds were tested in 10-dose IC50 triplicate mode with a 3-fold...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.935nMAssay Description:Inhibition of human PKA using LCGRTGRRNSI as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799597BDBM799597(US12583856, Example 106)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50117503BDBM50117503(CHEMBL3613621)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799598BDBM799598(US12583856, Example 107)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799599BDBM799599(US12583856, Example 108)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799600BDBM799600(US12583856, Example 109)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50117504BDBM50117504(CHEMBL3613620)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799601BDBM799601(US12583856, Example 110)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799604BDBM799604(US12583856, Example 111)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799607BDBM799607(US12583856, Example 112)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799478BDBM799478(US12583856, Example 100)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799480BDBM799480(US12583856, Example 101)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799487BDBM799487(US12583856, Example 102)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799504BDBM799504(US12583856, Example 103)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799594BDBM799594(US12583856, Example 104)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50044004BDBM50044004(CHEMBL3356433)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117489BDBM50117489(CHEMBL3613598)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799639BDBM799639(US12583856, Example 137)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799640BDBM799640(US12583856, Example 138)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799641BDBM799641(US12583856, Example 139)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799644BDBM799644(US12583856, Example 140)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799646BDBM799646(US12583856, Example 141)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799647BDBM799647(US12583856, Example 142)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799648BDBM799648(US12583856, Example 143)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799649BDBM799649(US12583856, Example 144)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799630BDBM799630(US12583856, Example 129)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799631BDBM799631(US12583856, Example 130)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799632BDBM799632(US12583856, Example 131)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799633BDBM799633(US12583856, Example 132)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799635BDBM799635(US12583856, Example 134)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799636BDBM799636(US12583856, Example 135)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799638BDBM799638(US12583856, Example 136)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799620BDBM799620(US12583856, Example 121)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799622BDBM799622(US12583856, Example 122)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799623BDBM799623(US12583856, Example 123)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799624BDBM799624(US12583856, Example 124)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799625BDBM799625(US12583856, Example 125)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799627BDBM799627(US12583856, Example 126)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 799628BDBM799628(US12583856, Example 127)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/3/2026
Entry Details
US Patent

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