Compile Data Set for Download or QSAR
maximum 50k data
Found 81 of affinity data for UniProtKB/TrEMBL: P20789
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]neurotensin from rat NTS1 receptor expressed in CHO-K1 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]neurotensin from rat NTS1 receptor expressed in CHO-K1 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  2nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50248034(2-{[1-(7-Chloro-quinolin-4-yl)-5-(2,6-dimethoxy-ph...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]NT from rat NTR1 transfected in mouse LTK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50041427(CHEMBL3356853)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50041429(CHEMBL3356854)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50041428(CHEMBL3356855)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366375(CHEMBL1794002)
Affinity DataKi:  29nMAssay Description:Tested for binding affinity against Neurotensin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281809((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-6-Amino-2-ter...)
Affinity DataKi:  63nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281809((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-6-Amino-2-ter...)
Affinity DataKi:  63nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281812((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-5-Amino-2-ter...)
Affinity DataKi:  82nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281812((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-5-Amino-2-ter...)
Affinity DataKi:  82nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366303(CHEMBL1790460)
Affinity DataKi:  100nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi:  117nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi:  120nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50019412(CHEMBL3290096)
Affinity DataKi:  177nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366296(CHEMBL1790463)
Affinity DataKi:  180nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366308(CHEMBL1790472)
Affinity DataKi:  190nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366299(CHEMBL1790467)
Affinity DataKi:  220nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366307(CHEMBL1790457)
Affinity DataKi:  290nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366298(CHEMBL1790466)
Affinity DataKi:  420nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366311(CHEMBL1790470)
Affinity DataKi:  520nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366302(CHEMBL2369587)
Affinity DataKi:  540nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366310(CHEMBL1790461)
Affinity DataKi:  680nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281807((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-2,6-Diamino-h...)
Affinity DataKi:  688nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281807((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-2,6-Diamino-h...)
Affinity DataKi:  690nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366371(CHEMBL1793833)
Affinity DataKi:  730nMAssay Description:Tested for binding affinity against Neurotensin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366300(CHEMBL1790465)
Affinity DataKi:  880nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366374(CHEMBL1793999)
Affinity DataKi:  890nMAssay Description:Tested for binding affinity against Neurotensin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366304(CHEMBL2369588)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50019417(CHEMBL3290101)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366370(CHEMBL1794003)
Affinity DataKi:  1.25E+3nMAssay Description:Tested for binding affinity against Neurotensin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281806((S)-2-{(2S,3S)-2-[(S)-2-{N'-[2-((S)-1-{(S)-2-[(Ada...)
Affinity DataKi:  1.61E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281810((S)-2-{(2S,3S)-2-[(S)-2-{(E)-3-[(S)-1-((S)-6-Amino...)
Affinity DataKi:  1.63E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366301(CHEMBL1790469)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366306(CHEMBL1790473)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366373(CHEMBL1794000)
Affinity DataKi:  2.20E+3nMAssay Description:Tested for binding affinity against Neurotensin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281804((S)-2-{(2S,3S)-2-[(S)-2-(N'-{2-[(S)-1-((S)-5-Amino...)
Affinity DataKi:  2.99E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50019423(CHEMBL3290105)
Affinity DataKi:  3.21E+3nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281813((S)-2-((2S,3S)-2-{N'-[(S)-3-[((S)-1-{(S)-3-[(Adama...)
Affinity DataKi:  3.86E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281805((S)-2-((2S,3S)-2-{N'-[(S)-3-[((S)-1-{(S)-2-[(Adama...)
Affinity DataKi:  5.96E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50069089(CHEMBL3403505)
Affinity DataKi:  7.18E+3nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366312(CHEMBL1790476)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50069088(CHEMBL3403504)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50366372(CHEMBL1793998)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for binding affinity against Neurotensin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50281808((S)-2-((2S,3S)-2-{N'-[(S)-3-{[(S)-1-((S)-5-Amino-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50069090(CHEMBL3403506)
Affinity DataKi:  1.02E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50069091(CHEMBL3403507)
Affinity DataKi: >2.50E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50069092(CHEMBL3403508)
Affinity DataKi: >2.50E+4nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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