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TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50122050(N-{2-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  0.0180nMAssay Description:Binding affinity towards human Dopamine receptor D4 using [3H]spiroperidol as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50122028(3-Methoxy-N-[2-(4-p-tolyl-piperazin-1-yl)-ethyl]-b...)
Affinity DataKi:  0.0250nMAssay Description:Binding affinity towards human Dopamine receptor D4 using [3H]spiroperidol as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50005120(Nemonapride | N-((2S,3S)-1-Benzyl-2-methyl-pyrroli...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2012
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50005120(Nemonapride | N-((2S,3S)-1-Benzyl-2-methyl-pyrroli...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2012
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50530438(Mosapramine | Mosapramine hydrochloride)
Affinity DataKi:  0.0300nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50530438(Mosapramine | Mosapramine hydrochloride)
Affinity DataKi:  0.0300nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50068366(N-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-3...)
Affinity DataKi:  0.0400nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]YM-09151-2 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50122026(N-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethyl}-3...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity towards human Dopamine receptor D4 using [3H]spiroperidol as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50068366(N-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-3...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity towards human Dopamine receptor D4 using [3H]spiroperidol as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50068366(N-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-3...)
Affinity DataIC50: 0.0570nMAssay Description:In vitro binding affinity at human cloned Dopamine receptor D4.2 by [3H]YM-09151-2 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM81492(CAS_2062-84-2 | NSC_16363 | BENPERIDOL)
Affinity DataKi:  0.0660nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50183266(Anquil | Benperidol | Benquil | MCN-JR-4584 | R-45...)
Affinity DataKi:  0.0660nMAssay Description:Binding affinity to human dopamine D4 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50568740(CHEMBL4860528)
Affinity DataKd:  0.0780nMAssay Description:Displacement of [3H]N-methylspiperone from human D4.4 receptor stably expressed in HEK293T cells co-expressing ElucN-betaarr2 hD4.4R-ELuc incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50601567(CHEMBL5206565)
Affinity DataKd:  0.0780nMAssay Description:Displacement of [3H]N-methylspiperone from human D4.4 receptor stably expressed in HEK293T cells co-expressing ElucN-betaarr2 hD4.4R-ELuc incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50601551(CHEMBL5207281)
Affinity DataKd:  0.0780nMAssay Description:Displacement of [3H]N-methylspiperone from human D4.4 receptor stably expressed in HEK293T cells co-expressing ElucN-betaarr2 hD4.4R-ELuc incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50601574(CHEMBL5201074)
Affinity DataKd:  0.0780nMAssay Description:Displacement of [3H]N-methylspiperone from human D4.4 receptor stably expressed in HEK293T cells co-expressing ElucN-betaarr2 hD4.4R-ELuc incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM85223(NSC_115368 | CAS_115368 | Perospirone)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50263488(CHEMBL4085780)
Affinity DataEC50:  0.158nMAssay Description:Agonist activity at human SP/Myc epitope-tagged dopamine D4 receptor expressed in HEK293T cells assessed as RLuc8-fused Galphai1 activation after 2 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50608795(CHEMBL5290993)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at D4R (unknown origin) by camp reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50005120(Nemonapride | N-((2S,3S)-1-Benzyl-2-methyl-pyrroli...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50454212(CHEBI:64217 | Emonapride | Nemonapride)
Affinity DataKd:  0.210nMAssay Description:Binding Affinity to Human Dopamine receptor D4 expressed in CHO cells was determined using [3H]- nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50122032(3-Methoxy-N-[2-(4-naphthalen-1-yl-piperazin-1-yl)-...)
Affinity DataKi:  0.210nMAssay Description:Binding affinity towards human Dopamine receptor D4 using [3H]spiroperidol as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM84637(NSC_54562 | CHEMBL240773 | QUINPIROLE | CAS_85760-...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2012
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.25nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50505700(CHEMBL4442460)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H] Spiperone from human D4.4 receptor expressed in CHO cells by competitive radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.25nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50122047(N-{2-[4-(3-Chloro-phenyl)-piperazin-1-yl]-ethyl}-3...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity towards human Dopamine receptor D4 using [3H]spiroperidol as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50184795(1-(2-methoxyphenyl)-4-((1-phenyl-1H-pyrazol-4-yl)m...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM85222(Lurasidone | CAS_441351-20-8 | SM 13496)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50061349([2-(3-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-am...)
Affinity DataKi:  0.309nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50061349([2-(3-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-am...)
Affinity DataKi:  0.310nMAssay Description:Binding affinity to recombinant human dopamine receptor D4 expressed in CHO cells by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity for Dopamine receptor D4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.330nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  0.330nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50079161(5-Methyl-1-[1-(3-methyl-benzyl)-piperidin-4-yl]-4-...)
Affinity DataKi:  0.330nMAssay Description:Affinity to displace [3H]spiperone from cloned human Dopamine receptor D4 stably expressed in HEK393 cell linesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.330nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]-spiperone from D4 (unknown origin) receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  0.331nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50061345([2-(3,4-Dimethyl-phenoxy)-ethyl]-(3-phenoxy-propyl...)
Affinity DataKi:  0.347nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM81493(CAS_749-13-3 | TRIFLUORPERIDOL)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50061345([2-(3,4-Dimethyl-phenoxy)-ethyl]-(3-phenoxy-propyl...)
Affinity DataKi:  0.350nMAssay Description:Binding affinity to recombinant human dopamine receptor D4 expressed in CHO cells by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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