Compile Data Set for Download or QSAR
maximum 50k data
Found 1251 of affinity data for UniProtKB/TrEMBL: P47900
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50373326(CHEMBL444278)
Affinity DataKi:  0.780nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50373326(CHEMBL444278)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]2-chloro-N 6- methyl-( N )-methanocarba-2'-deoxyadenosine 3 ' ,5 '-bis-phosphate from human P2Y1 expressed in baculovirus infecte...More data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50373326(CHEMBL444278)
Affinity DataKi:  0.780nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM261048(US9540323, 269 | US9540323, example 269)
Affinity DataKi:  1.20nM ΔG°:  -50.9kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245383(US9428504, 133)
Affinity DataKi:  1.20nM ΔG°:  -50.9kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245297(US9428504, 35)
Affinity DataKi:  1.90nM ΔG°:  -49.8kJ/moleT: 2°CAssay Description:Binding reactions were performed in WGA FLASHPLATEs (PerkinElmer Life Sciences, Cat # SMP105A) in a volume of 200 uL containing 45 fmol of P2Y1 recep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50409757(CHEMBL2112864)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260841(US9540323, 27 | US9540323, example 27)
Affinity DataKi:  3.10nM ΔG°:  -48.6kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245282(US9428504, 20)
Affinity DataKi:  3.20nM ΔG°:  -48.5kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015276(CHEMBL3263056 | US9428504, 166 | US9428504, 167)
Affinity DataKi:  3.30nM ΔG°:  -48.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245275(US9428504, 13)
Affinity DataKi:  3.30nM ΔG°:  -48.4kJ/moleT: 2°CAssay Description:Binding reactions were performed in WGA FLASHPLATEs (PerkinElmer Life Sciences, Cat # SMP105A) in a volume of 200 uL containing 45 fmol of P2Y1 recep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260928(US9540323, 119 | US9540323, example 119)
Affinity DataKi:  3.30nM ΔG°:  -48.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245302(US9428504, 42)
Affinity DataKi:  3.30nM ΔG°:  -48.4kJ/moleT: 2°CAssay Description:Binding reactions were performed in WGA FLASHPLATEs (PerkinElmer Life Sciences, Cat # SMP105A) in a volume of 200 uL containing 45 fmol of P2Y1 recep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260845(US9540323, 31 | US9540323, example 31)
Affinity DataKi:  3.30nM ΔG°:  -48.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260816(US9540323, 2 | US9540323, example 2)
Affinity DataKi:  3.40nM ΔG°:  -48.3kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260932(US9540323, 124 | US9540323, example 124)
Affinity DataKi:  3.40nM ΔG°:  -48.3kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245342(US9428504, 91)
Affinity DataKi:  3.40nM ΔG°:  -48.3kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245341(US9428504, 90)
Affinity DataKi:  3.5nM ΔG°:  -48.3kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50409764(CHEMBL2112867)
Affinity DataKi:  3.60nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260843(US9540323, 29 | US9540323, example 29)
Affinity DataKi:  3.60nM ΔG°:  -48.2kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245295(US9428504, 33)
Affinity DataKi:  3.70nM ΔG°:  -48.1kJ/moleT: 2°CAssay Description:Binding reactions were performed in WGA FLASHPLATEs (PerkinElmer Life Sciences, Cat # SMP105A) in a volume of 200 uL containing 45 fmol of P2Y1 recep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245296(US9428504, 34)
Affinity DataKi:  3.70nM ΔG°:  -48.1kJ/moleT: 2°CAssay Description:Binding reactions were performed in WGA FLASHPLATEs (PerkinElmer Life Sciences, Cat # SMP105A) in a volume of 200 uL containing 45 fmol of P2Y1 recep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245340(US9428504, 85)
Affinity DataKi:  3.70nM ΔG°:  -48.1kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50017083(CHEMBL3287049 | US9428504, 39)
Affinity DataKi:  3.80nM ΔG°:  -48.1kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245414(US9428504, 173)
Affinity DataKi:  3.80nM ΔG°:  -48.1kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50017021(CHEMBL3287047 | US9428504, 1)
Affinity DataKi:  4nMAssay Description:Binding affinity to P2Y1 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245271(US9428504, 7)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260870(US9540323, 58 | US9540323, example 58)
Affinity DataKi:  4.10nM ΔG°:  -47.9kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260934(US9540323, 126 | US9540323, example 126)
Affinity DataKi:  4.10nM ΔG°:  -47.9kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50445214(CHEMBL3104636)
Affinity DataKi:  4.30nMAssay Description:Displacement of [33P]-2MeS-ADP from human P2Y1 receptor expressed in HEK293 cells after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245284(US9428504, 22)
Affinity DataKi:  4.40nM ΔG°:  -47.7kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245303(US9428504, 43)
Affinity DataKi:  4.40nM ΔG°:  -47.7kJ/moleT: 2°CAssay Description:Binding reactions were performed in WGA FLASHPLATEs (PerkinElmer Life Sciences, Cat # SMP105A) in a volume of 200 uL containing 45 fmol of P2Y1 recep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50017091(CHEMBL3287045 | US9428504, 6)
Affinity DataKi:  4.40nM ΔG°:  -47.7kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260885(US9540323, 73 | US9540323, example 73)
Affinity DataKi:  4.5nM ΔG°:  -47.6kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50017087(CHEMBL3287041 | US9428504, 10)
Affinity DataKi:  4.5nM ΔG°:  -47.6kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260931(US9540323, 123 | US9540323, example 123)
Affinity DataKi:  4.5nM ΔG°:  -47.6kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50045627(CHEMBL3314307 | US9540323, 200 | US9540323, exampl...)
Affinity DataKi:  4.60nM ΔG°:  -47.6kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50445208(CHEMBL3105199)
Affinity DataKi:  4.60nMAssay Description:Displacement of [33P]-2MeS-ADP from human P2Y1 receptor expressed in HEK293 cells after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260935(US9540323, 127 | US9540323, example 127)
Affinity DataKi:  4.70nM ΔG°:  -47.5kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260987(US9540323, 188 | US9540323, example 188)
Affinity DataKi:  4.70nM ΔG°:  -47.5kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260933(US9540323, 125 | US9540323, example 125)
Affinity DataKi:  4.80nM ΔG°:  -47.5kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245320(US9428504, 63)
Affinity DataKi:  4.90nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260996(US9540323, 212 | US9540323, example 212)
Affinity DataKi:  4.90nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50045625(CHEMBL3314305 | US9540323, 198 | US9540323, exampl...)
Affinity DataKi:  4.90nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245287(US9428504, 25)
Affinity DataKi:  4.90nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260817(US9540323, 3 | US9540323, example 3)
Affinity DataKi:  4.90nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM260826(US9540323, 12 | US9540323, example 12)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50436912(CHEMBL2401804)
Affinity DataKi:  5nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 expressed in HEK293 cells after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM245336(US9428504, 81)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50436912(CHEMBL2401804)
Affinity DataKi:  5nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor expressed in HEK293 cells after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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