Affinity DataIC50: 59nMAssay Description:Inhibition of KHK in mouse hepatocytes using D-fructose as substrate assessed as reduction in fructose-1-phosphate level preincubated for 30 mins fol...More data for this Ligand-Target Pair
Affinity DataEC50: 134nMAssay Description:Experiment of Inhibitory Activity Against KHK In Vitro: With the involvement of ATP, fructokinase phosphorylates fructose to produce fructose-1-phosp...More data for this Ligand-Target Pair

3D Structure (crystal)