Affinity DataIC50: 3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 129nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Allosteric modulation of mouse PDE4DMore data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 220nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 323nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 653nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.68E+3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 5.91E+3nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
TargetPhosphodiesterase/cAMP-specific 3',5'-cyclic phosphodiesterase 4A/cAMP-specific 3',5'-cyclic phosphodiesterase 4C/cAMP-specific 3',5'-cyclic phosphodiesterase 4D(Mus musculus)TBA
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair