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Report error Found 760 of affinity data for UniProtKB/TrEMBL: Q13043
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM21079(1-[4-(3-azanyl-1H-indazol-4-yl)phenyl]-3-(2-fluora...)
Affinity DataKd:  1.40E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM25118(4-amino-5-fluoro-3-[6-(4-methylpiperazin-1-yl)-1H-...)
Affinity DataKd:  200nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-etho...)
Affinity DataKd:  3.60E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM6866(1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3b ...)
Affinity DataKd:  130nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31094(PKC-412 | cid_24202429)
Affinity DataKd:  40nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd:  130nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705 | US2024...)
Affinity DataKd:  0.190nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  19nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM13534(VX680 | N-[4-[[4-(4-methylpiperazino)-6-[(5-methyl...)
Affinity DataKd:  200nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50505541(CHEMBL4465866)
Affinity DataKd:  7nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged STK4 (unknown origin) expressed in baculovirus infected Sf9 insect cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50505542(CHEMBL4576489)
Affinity DataKd:  4nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged STK4 (unknown origin) expressed in baculovirus infected Sf9 insect cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50059345(CHEMBL3393355 | US9156845, 83 | US20250051337, Com...)
Affinity DataKd:  147nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human STK4 (43 to 431 residues) expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50583973(CHEMBL5093114 | US20250051337, Compound 23)
Affinity DataKd:  158nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human STK4 (43 to 431 residues) expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50024294(SP-600125)
Affinity DataKd:  2.20E+3nMAssay Description:Average Binding Constant for STK4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  0.200nMAssay Description:Average Binding Constant for STK4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM17055((9S)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydr...)
Affinity DataKd:  220nMAssay Description:Average Binding Constant for STK4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  100nMAssay Description:Average Binding Constant for STK4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-etho...)
Affinity DataKd:  3.90E+3nMAssay Description:Average Binding Constant for STK4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50599287(CHEMBL5183592 | US12318398, Compound 25)
Affinity DataKd:  240nMAssay Description:Binding affinity to wild-type human full length MST1 (M1 to F487 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  1nMAssay Description:Binding affinity to recombinant STK4 (unknown origin) assessed as dissociation constant by DSF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50148921(CHEMBL3770443)
Affinity DataEC50:  3.04E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641138(CHEMBL5592121)
Affinity DataEC50:  1.28E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641139(CHEMBL5574332)
Affinity DataEC50:  3.14E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641140(CHEMBL5592254)
Affinity DataEC50:  9.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641141(CHEMBL5572457)
Affinity DataEC50:  5.30E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641142(CHEMBL5572173)
Affinity DataEC50:  7.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641143(CHEMBL5556031)
Affinity DataEC50:  6.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641144(CHEMBL5589642)
Affinity DataEC50:  3.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641145(CHEMBL5566862)
Affinity DataEC50:  3.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641146(CHEMBL5569169)
Affinity DataEC50: >5.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50182295(CHEMBL3818046)
Affinity DataEC50:  2.63E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641147(CHEMBL5567421)
Affinity DataEC50:  4.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641148(CHEMBL5567287)
Affinity DataEC50:  2.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641149(CHEMBL5555859)
Affinity DataEC50:  1.60E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641150(CHEMBL5575508)
Affinity DataEC50:  660nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataEC50:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641151(CHEMBL5573797)
Affinity DataEC50: >5.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641152(CHEMBL5572995)
Affinity DataEC50:  3.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641153(CHEMBL5565155)
Affinity DataEC50:  5.30E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641154(CHEMBL5566570)
Affinity DataEC50:  1.51E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641155(CHEMBL5572984)
Affinity DataEC50:  5.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641156(CHEMBL5590480)
Affinity DataEC50: >5.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641157(CHEMBL5571159)
Affinity DataEC50:  251nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641158(CHEMBL5569777)
Affinity DataEC50:  419nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641159(CHEMBL5594538)
Affinity DataEC50:  530nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641160(CHEMBL5571948)
Affinity DataEC50:  314nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641161(CHEMBL5590631)
Affinity DataEC50:  3.30E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641162(CHEMBL5573230)
Affinity DataEC50:  2.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50641163(CHEMBL5567028)
Affinity DataEC50: >5.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetSerine/threonine-protein kinase 4(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50613306(CHEMBL1235645)
Affinity DataEC50:  200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
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