Compile Data Set for Download or QSAR
maximum 50k data
Found 45 of affinity data for UniProtKB/TrEMBL: Q8BGY9
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416502(CHEMBL1209654)
Affinity DataKi:  20.0nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416489(CHEMBL1209507)
Affinity DataKi:  50nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416490(CHEMBL1209508)
Affinity DataKi:  90.0nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416491(CHEMBL1209577)
Affinity DataKi:  180nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416508(CHEMBL1209578)
Affinity DataKi:  200nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416504(CHEMBL1209579)
Affinity DataKi:  230nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416506(CHEMBL1209581)
Affinity DataKi:  521nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416503(CHEMBL1209713)
Affinity DataKi:  640nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026220(2-hydroxy-N,N,N-trimethylethanaminium | CHEMBL2824...)
Affinity DataKi:  681nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416501(CHEMBL1209653)
Affinity DataKi:  701nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416488(CHEMBL1209506)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50147119((3-Hydroxy-propyl)-trimethyl-ammonium | CHEMBL1209...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50204415(1-methyl-1-azonia-bicyclo[2.2.2]octane | CHEMBL120...)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50079455(CHEMBL46486 | tetramethylammonium)
Affinity DataKi:  3.01E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM80992(1-cetylpyridin-1-ium;bromide | 1-hexadecylpyridin-...)
Affinity DataKi:  3.21E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416495(CHEMBL1209648)
Affinity DataKi:  4.01E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060526(2-Dimethylamino-ethanol | 2-hydroxy-N,N-dimethylet...)
Affinity DataKi:  5.57E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416507(CHEMBL1209649)
Affinity DataKi:  7.21E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM80386(CHEMBL1209421 | MLS000069658 | PHENYLTRIMETHYLAMMO...)
Affinity DataKi:  7.52E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416505(CHEMBL1209580)
Affinity DataKi:  1.07E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416484(CHEMBL1209503)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416496(CHEMBL1209650)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50047005(1-Aza-bicyclo[2.2.2]octan-3-ol | 1-Aza-bicyclo[2.2...)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416485(CHEMBL1209504)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416483(CHEMBL1209424)
Affinity DataKi:  2.90E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50147105((4-Hydroxy-butyl)-trimethyl-ammonium | CHEMBL10228...)
Affinity DataKi:  3.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416486(CHEMBL1209505)
Affinity DataKi:  3.40E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416499(TRIMETHYLAMMONIUM)
Affinity DataKi:  3.40E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416500(CHEMBL1209652)
Affinity DataKi:  3.61E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM10458(4-AP | 4-Aminopyridine 10 | CHEMBL284348 | DALFAMP...)
Affinity DataKi:  4.81E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416493(CHEMBL354077)
Affinity DataKi:  8.20E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataKi:  1.05E+6nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50147120(2-Methylamino-ethanol | 2-hydroxy-N-methylethanami...)
Affinity DataKi:  3.80E+6nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416497(DIMETHYLAMINE)
Affinity DataKi:  9.42E+6nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416492(Integrase inhibitor, R3{3} | METHYLAMINE)
Affinity DataKi:  3.51E+7nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM7973(2-aminoethan-1-ol | CHEMBL104943 | ethanolamine)
Affinity DataKi:  1.50E+8nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026216(1-Ethyl-1-(2-hydroxy-ethyl)-aziridinium; chloride ...)
Affinity DataIC50:  1.50E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026220(2-hydroxy-N,N,N-trimethylethanaminium | CHEMBL2824...)
Affinity DataIC50:  1.60E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026218(1-(2-Hydroxy-ethyl)-1-isopropyl-aziridinium; chlor...)
Affinity DataIC50:  2.60E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026215(1-Cyclopropyl-1-(2-hydroxy-ethyl)-aziridinium; chl...)
Affinity DataIC50:  3.90E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026219(1-(2-Hydroxy-ethyl)-1-propyl-aziridinium; chloride...)
Affinity DataIC50:  7.50E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026217(1-(2-Hydroxy-ethyl)-1-isobutyl-aziridinium; chlori...)
Affinity DataIC50:  3.10E+4nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026221(1-Butyl-1-(2-hydroxy-ethyl)-aziridinium; chloride ...)
Affinity DataIC50: >1.00E+6nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed