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Found 1064 of affinity data for UniProtKB/TrEMBL: Q96S37
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50538736(CHEMBL4640580)
Affinity DataKi:  57nMAssay Description:Inhibition of human URAT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM26658(2-(2,4-dihydroxyphenyl)-3,5,7-trihydroxy-1-benzopy...)
Affinity DataKi:  5.74E+3nMAssay Description:Inhibition of human URAT1-mediated urate uptake in HEK293 cells by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM165905(US9067922, 247)
Affinity DataIC50:  1nMpH: 7.4Assay Description:Assay compound plates were prepared by diluting the compounds of formula (I) with chloride-free buffer (125 mM Na-gluconate, 4.8 mM K-gluconate, 1.3 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50239134(CHEMBL4087516)
Affinity DataIC50:  2nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells assessed as reduction in [14C]uric acid uptake measured after 5 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM165898(US9067922, 239)
Affinity DataIC50:  2nMpH: 7.4Assay Description:Assay compound plates were prepared by diluting the compounds of formula (I) with chloride-free buffer (125 mM Na-gluconate, 4.8 mM K-gluconate, 1.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM165900(US9067922, 241)
Affinity DataIC50:  3nMpH: 7.4Assay Description:Assay compound plates were prepared by diluting the compounds of formula (I) with chloride-free buffer (125 mM Na-gluconate, 4.8 mM K-gluconate, 1.3 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612481(CHEMBL5271398)
Affinity DataIC50:  3.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50546900(CHEMBL4756866)
Affinity DataIC50:  4.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM165745(US9067922, 235 | US9067922, 79)
Affinity DataIC50:  7nMpH: 7.4Assay Description:Assay compound plates were prepared by diluting the compounds of formula (I) with chloride-free buffer (125 mM Na-gluconate, 4.8 mM K-gluconate, 1.3 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612476(CHEMBL5277301)
Affinity DataIC50:  7.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612472(CHEMBL5284974)
Affinity DataIC50:  7.60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612468(CHEMBL5287151)
Affinity DataIC50:  7.70nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612477(CHEMBL5289202)
Affinity DataIC50:  7.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM290450(2{[4-(4-Cyanonaphthalen)isoquinolin-6-yl]thio}-2-m...)
Affinity DataIC50:  8nMAssay Description:Human embryonic kidney cells (HEK293) was incubated in DMEM tissue culture medium, at 37° C., under 5% CO2 and 95% air atmosphere. TransIT-293 transf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM165896(US9067922, 237)
Affinity DataIC50:  8nMpH: 7.4Assay Description:Assay compound plates were prepared by diluting the compounds of formula (I) with chloride-free buffer (125 mM Na-gluconate, 4.8 mM K-gluconate, 1.3 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612478(CHEMBL5269373)
Affinity DataIC50:  9.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM37953(US10093631, Compound Lesinurad | US10336710, Lesin...)
Affinity DataIC50:  9.40nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612475(CHEMBL5278085)
Affinity DataIC50:  9.70nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612464(CHEMBL5279672)
Affinity DataIC50:  9.70nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612485(CHEMBL5289441)
Affinity DataIC50:  9.80nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612465(CHEMBL5273217)
Affinity DataIC50:  9.80nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612469(CHEMBL5277066)
Affinity DataIC50:  9.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612488(CHEMBL5290258)
Affinity DataIC50:  10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612490(CHEMBL5268478)
Affinity DataIC50:  10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50239146(CHEMBL4088988)
Affinity DataIC50:  10nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells assessed as reduction in [14C]uric acid uptake measured after 5 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM290480(US10100016, Compound 45B)
Affinity DataIC50:  10nMAssay Description:Human embryonic kidney cells (HEK293) was incubated in DMEM tissue culture medium, at 37° C., under 5% CO2 and 95% air atmosphere. TransIT-293 transf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM152041(US8987473, 122)
Affinity DataIC50:  10nMAssay Description:It was introduced human URAT1 full-length cDNA into an expression vector pcDNA5 / FRT / V5-His TOPO (registered trademark) (Invitrogen). The result...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM152051(US8987473, 137)
Affinity DataIC50:  10nMAssay Description:It was introduced human URAT1 full-length cDNA into an expression vector pcDNA5 / FRT / V5-His TOPO (registered trademark) (Invitrogen). The result...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612470(CHEMBL5291373)
Affinity DataIC50:  11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612479(CHEMBL5285786)
Affinity DataIC50:  11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612482(CHEMBL5282615)
Affinity DataIC50:  11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612491(CHEMBL5267727)
Affinity DataIC50:  11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612463(CHEMBL5267010)
Affinity DataIC50:  11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM290470(US10100016, Compound 43A)
Affinity DataIC50:  11nMAssay Description:Human embryonic kidney cells (HEK293) was incubated in DMEM tissue culture medium, at 37° C., under 5% CO2 and 95% air atmosphere. TransIT-293 transf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612466(CHEMBL5285533)
Affinity DataIC50:  12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612471(CHEMBL5282586)
Affinity DataIC50:  12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612480(CHEMBL5268476)
Affinity DataIC50:  12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612487(CHEMBL5290341)
Affinity DataIC50:  12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612493(CHEMBL5266247)
Affinity DataIC50:  12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM290481(3-[4-(4-Cyanonaphthalen-1-yl)isoquinolin-6-yl]-2,2...)
Affinity DataIC50:  12nMAssay Description:Human embryonic kidney cells (HEK293) was incubated in DMEM tissue culture medium, at 37° C., under 5% CO2 and 95% air atmosphere. TransIT-293 transf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM290489(3-[4-(4-Cyanophenyl)thieno[2,3-c]pyridin-2-yl]-2,2...)
Affinity DataIC50:  12nMAssay Description:Human embryonic kidney cells (HEK293) was incubated in DMEM tissue culture medium, at 37° C., under 5% CO2 and 95% air atmosphere. TransIT-293 transf...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM318948(2-Methyl-2-[[7-(4-nitrophenyl)benzo[d]isothiazol-6...)
Affinity DataIC50:  12nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM165893(US9067922, 232)
Affinity DataIC50:  12nMpH: 7.4Assay Description:Assay compound plates were prepared by diluting the compounds of formula (I) with chloride-free buffer (125 mM Na-gluconate, 4.8 mM K-gluconate, 1.3 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612474(CHEMBL5272958)
Affinity DataIC50:  13nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM165667(US9067922, 1)
Affinity DataIC50:  13nMpH: 7.4Assay Description:Assay compound plates were prepared by diluting the compounds of formula (I) with chloride-free buffer (125 mM Na-gluconate, 4.8 mM K-gluconate, 1.3 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM165745(US9067922, 235 | US9067922, 79)
Affinity DataIC50:  13nMpH: 7.4Assay Description:Assay compound plates were prepared by diluting the compounds of formula (I) with chloride-free buffer (125 mM Na-gluconate, 4.8 mM K-gluconate, 1.3 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM152048(US8987473, 134)
Affinity DataIC50:  13nMAssay Description:It was introduced human URAT1 full-length cDNA into an expression vector pcDNA5 / FRT / V5-His TOPO (registered trademark) (Invitrogen). The result...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612486(CHEMBL5278304)
Affinity DataIC50:  14nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM377700(US10266496, Example 27)
Affinity DataIC50:  14nMAssay Description:a. Construction of a Cell Line Stably Expressing hURAT1hURAT1 plasmid was transfected into HEK293T cell, and a cell line stably expressing hURAT1 was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
West China Hospital Of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50612492(CHEMBL5272326)
Affinity DataIC50:  15nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
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