TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of RIOK2 in human VCaP cells after 48 hrs by Western blotting analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 139nMAssay Description:Inhibition of N-terminal hexahistidine-SUMO-tagged human full length RIOK2 (residues 1 to 321) expressed in Escherichia coli BL21 (DE3) incubated for...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: <5.89E+3nMAssay Description:Inhibition of RIOK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of fluorescent tracer K5 from N-terminal full-length NanoLuc-fused RIOK2 (unknown origin) expressed in HEK293 cells using NanoGlo substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.34E+4nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.45E+4nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.46E+4nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.46E+4nMAssay Description:Displacement of fluorescent tracer K5 from N-terminal full-length NanoLuc-fused RIOK2 (unknown origin) expressed in HEK293 cells using NanoGlo substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 6.70E+3nMAssay Description:Binding affinity to RIOK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 97nMAssay Description:Binding affinity to RIOK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 6.70E+3nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 97nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 390nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to RIOK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 49nMAssay Description:Binding affinity to RIOK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to RIOK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to RIOK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to RIOK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 2.60E+3nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: 770nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase RIO2(Homo sapiens (Human))
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Uniformed Services University Of The Health Sciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RIOK2 kinase domainMore data for this Ligand-Target Pair