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Report error Found 208 of affinity data for UniProtKB/TrEMBL: Q9BZL6
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human PKD2 using KKLNRTLSVA as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human PKD2 using KKLNRTLSVA as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM130909(US8822500, Stauro- sporine | US9920060, Staurospor...)
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM519645(US11142525, Example 46 | US11684616, Example 300)
Affinity DataIC50: 1.93nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50616058(CHEMBL5419827)
Affinity DataIC50: 2nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50616060(CHEMBL5428541)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606195(US11684616, Example 201)
Affinity DataIC50: 5.43nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606196(US11684616, Example 202)
Affinity DataIC50: 6.54nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606100(US11684616, Example 3)
Affinity DataIC50: 6.54nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606194(US11684616, Example 200)
Affinity DataIC50: 7.97nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd:  8.10nMAssay Description:Binding affinity to PRKD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd:  8.10nMAssay Description:Binding constant for PRKD2 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50616054(CHEMBL5440043)
Affinity DataIC50: 9nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50565693(CHEMBL4515390)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50542119(CHEMBL4644939)
Affinity DataIC50: 17nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM101618(US8530652, 114)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM101618(US8530652, 114)
Affinity DataIC50: 26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  31nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50565690(CHEMBL4787572)
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50565692(CHEMBL4790321)
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM416549(US10307425, Example 15 | US10632122, Example 15)
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50337694((R)-N-(1-cyanoethyl)-3-(5-(4-((tetrahydro-2H-pyran...)
Affinity DataIC50: 48nMAssay Description:Inhibition of human PKD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606137(US11684616, Example 100)
Affinity DataIC50: 51.2nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50565691(CHEMBL4776166)
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50336960(kb-NB142-70 | CHEMBL1672571 | 3,4-Dihydro-9-hydrox...)
Affinity DataIC50: 58.7nMpH: 7.5 T: 2°CAssay Description:In vitro radiometric kinase assay were conducted using PKD1 from Biomol International, PKD2 from SignalChem and PKD3 Enzo Life Sciences.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50336960(kb-NB142-70 | CHEMBL1672571 | 3,4-Dihydro-9-hydrox...)
Affinity DataIC50: 59nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705 | US2024...)
Affinity DataKd:  72nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  72nMAssay Description:Binding constant for PRKD2 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  72nMAssay Description:Binding constant for PRKD2 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 72nMAssay Description:Competitive inhibition of PKD2 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50505541(CHEMBL4465866)
Affinity DataKd:  79nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-tagged PRKD2 (unknown origin) expressed in baculovirus infected Sf9 insect cells incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50565687(CHEMBL4779081)
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50204834(2-(5-chloro-2-fluorophenyl)-N-(pyridin-4-yl)pterid...)
Affinity DataIC50: 94nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50336962(CHEMBL1672573 | kb-NB165-92 | 2,3,4,5-Tetrahydro-1...)
Affinity DataIC50: 101nMpH: 7.5 T: 2°CAssay Description:In vitro radiometric kinase assay were conducted using PKD1 from Biomol International, PKD2 from SignalChem and PKD3 Enzo Life Sciences.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50542117(CHEMBL4640042)
Affinity DataIC50: 102nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606099(US11684616, Example 2)
Affinity DataIC50: 116nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50229961(1-(1,1-dimethylethyl)-3-(1-naphthalenyl)-1H-pyrazo...)
Affinity DataIC50: 133nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50360301(CHEMBL1933288 | US9150577, 93)
Affinity DataIC50: 139nMAssay Description:Inhibition of human PRKD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50505542(CHEMBL4576489)
Affinity DataKd:  140nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-tagged PRKD2 (unknown origin) expressed in baculovirus infected Sf9 insect cells incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50119286(CHEMBL319170 | PD-146626 | kb-NB165-09 | 3-Methoxy...)
Affinity DataIC50: 142nMpH: 7.5 T: 2°CAssay Description:In vitro radiometric kinase assay were conducted using PKD1 from Biomol International, PKD2 from SignalChem and PKD3 Enzo Life Sciences.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50542123(CHEMBL4636488)
Affinity DataIC50: 144nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606098(US11684616, Example 1)
Affinity DataIC50: 155nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM482158(TAE684 | BDBM50242742)
Affinity DataKd:  160nMAssay Description:Binding constant for PRKD2 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM81614(kb-NB165-31)
Affinity DataIC50: 163nMpH: 7.5 T: 2°CAssay Description:In vitro radiometric kinase assay were conducted using PKD1 from Biomol International, PKD2 from SignalChem and PKD3 Enzo Life Sciences.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50542118(CHEMBL4645229)
Affinity DataIC50: 187nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50542125(CHEMBL4643470)
Affinity DataIC50: 202nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606101(US11684616, Example 4)
Affinity DataIC50: 217nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM185148(BMS-690514 | (3R,4R)-4-amino-1-[[4-(3-methoxyanili...)
Affinity DataKd: <225nMAssay Description:Binding affinity to wild-type human partial length PRKD2 (A519 to E838 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50542116(CHEMBL4646995)
Affinity DataIC50: 246nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM606102(US11684616, Example 5)
Affinity DataIC50: 251nMAssay Description:PRKD2 (PKD2) and RPS6KA2 (RSK3) kinase assays were performed with Km-levels of ATP at the Thermo Fisher Scientific, Inc. (Madison, Wis.), using their...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2023
Entry Details
Go to US Patent

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