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Found 32 of affinity data for UniProtKB/TrEMBL: Q9NY47
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50164279((S)-3-(aminomethyl)-5-methylhexanoic acid | (S)-3-...)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]-gabapentin from human Cav alpha2delta2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50557449(CHEMBL4744000)
Affinity DataKi:  2.15E+3nMAssay Description:Displacement of [3H]-gabapentin from human Cav alpha2delta2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM436318(2-(ethylamino)-9- methyl-6-(3-(5-methyl- 1,3,4-oxa...)
Affinity DataKi:  2.97E+3nMAssay Description:Displacement of [3H]-gabapentin from human Cav alpha2delta2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM436321(9-methyl-6-(3-(5- methyl-1,3,4- oxadiazol-2-yl)phe...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-gabapentin from human Cav alpha2delta2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM436247(9-methyl-6-(3-(5- methyl-1,3,4- oxadiazol-2- yl)ph...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-gabapentin from human Cav alpha2delta2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM388642(Reboxe- tine | US9944618, Compound ID No. 178)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-gabapentin from human Cav alpha2delta2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348465(CHEMBL1801177)
Affinity DataIC50:  10nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348456(CHEMBL1801206)
Affinity DataIC50:  22nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348457(CHEMBL1801207)
Affinity DataIC50:  59nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348467(CHEMBL1801179)
Affinity DataIC50:  79nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348474(CHEMBL1801186)
Affinity DataIC50:  85nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348468(CHEMBL1801180)
Affinity DataIC50:  126nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348478(CHEMBL1801205)
Affinity DataIC50:  158nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348455(CHEMBL1801192)
Affinity DataIC50:  200nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348471(CHEMBL1801183)
Affinity DataIC50:  316nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348464(CHEMBL1801176)
Affinity DataIC50:  398nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348470(CHEMBL1801182)
Affinity DataIC50:  398nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348458(CHEMBL1801208)
Affinity DataIC50:  537nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348453(CHEMBL1801188)
Affinity DataIC50:  631nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348472(CHEMBL1801184)
Affinity DataIC50:  631nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348473(CHEMBL1801185)
Affinity DataIC50:  794nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348475(CHEMBL1801187)
Affinity DataIC50:  794nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348459(CHEMBL1801209)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348463(CHEMBL1801213)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348461(CHEMBL1801211)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348462(CHEMBL1801212)
Affinity DataIC50:  1.07E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348466(CHEMBL1801178)
Affinity DataIC50:  1.59E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348469(CHEMBL1801181)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348476(CHEMBL1801189)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348460(CHEMBL1801210)
Affinity DataIC50:  2.13E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348454(CHEMBL1801191)
Affinity DataIC50:  3.98E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-2(Homo sapiens (Human))
Esteve Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50348477(CHEMBL1801190)
Affinity DataIC50:  6.31E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed