Compile Data Set for Download or QSAR
Report error Found 53 of affinity data for UniProtKB/TrEMBL: Q9QUQ5
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666590BDBM50666590(CHEMBL6174203)
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666593BDBM50666593(CHEMBL6175169)
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666596BDBM50666596(CHEMBL6175851)
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666598BDBM50666598(CHEMBL6173536)
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666597BDBM50666597(CHEMBL6162804)
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666599BDBM50666599(CHEMBL6177854)
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50519473BDBM50519473(CHEMBL4546097)
Affinity DataIC50: 17nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666600BDBM50666600(CHEMBL6169683)
Affinity DataIC50: 28nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79626BDBM79626(2-(azepan-1-yl)-4,6-dimethylquinoline;2,2,2-triflu...)
Affinity DataIC50: 900nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77617BDBM77617(4-methyl-2-(1-piperidinyl)quinoline | cid_230710 |...)
Affinity DataIC50: 960nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced intracellular calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50519463BDBM50519463(CHEMBL4532004)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse TRPC4 expressed in HEK293 cells coexpressing M5 receptor assessed as reduction in TRPC4-mediated calcium influx by fluorescence m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79629BDBM79629(VU0206683-4 | 2-(azepan-1-yl)-6-fluoro-4-methylqui...)
Affinity DataIC50: 1.63E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79628BDBM79628(VU0204326-4 | 2-(azepan-1-yl)-4-methyl-quinoline;2...)
Affinity DataIC50: 1.96E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77625BDBM77625(cid_46891900 | VU0419900-1 | 6-ethyl-4-methyl-2-py...)
Affinity DataIC50: 2.05E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 72595BDBM72595(2-(azepan-1-yl)-7-methoxy-4-methylquinoline;oxalic...)
Affinity DataIC50: 2.38E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77617BDBM77617(4-methyl-2-(1-piperidinyl)quinoline | cid_230710 |...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced current by QPatch cl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77617BDBM77617(4-methyl-2-(1-piperidinyl)quinoline | cid_230710 |...)
Affinity DataIC50: 2.63E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77618BDBM77618(4-methyl-2-(4-methyl-1-piperidinyl)quinoline;2,2,2...)
Affinity DataIC50: 3.14E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79627BDBM79627(VU0424395-1 | 2-(azepan-1-yl)-6-ethyl-4-methyl-qui...)
Affinity DataIC50: 3.30E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77620BDBM77620(4-methyl-2-pyrrolidin-1-ylquinoline;2,2,2-trifluor...)
Affinity DataIC50: 3.59E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492279BDBM50492279(CHEMBL1376358)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced intracellular calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77624BDBM77624(4,6-dimethyl-2-pyrrolidin-1-ylquinoline;2,2,2-trif...)
Affinity DataIC50: 3.71E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79623BDBM79623(VU0419899-1 | cid_46891898 | 6-ethyl-4-methyl-2-(1...)
Affinity DataIC50: 3.73E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79624BDBM79624(6-fluoro-4-methyl-2-pyrrolidin-1-ylquinoline;2,2,2...)
Affinity DataIC50: 3.94E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50519474BDBM50519474(CHEMBL4436705)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77621BDBM77621(VU0418910-1 | 4-methyl-2-[(2S)-2-methylpyrrolidin-...)
Affinity DataIC50: 4.26E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77614BDBM77614(SMR000122006 | MLS000529531 | 5-(4-fluorophenyl)-N...)
Affinity DataIC50: 4.28E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492273BDBM50492273(CHEMBL2396913)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77616BDBM77616(SMR000293019 | 4-chloro-N-cyclohexylbenzenecarboxi...)
Affinity DataIC50: 4.56E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239167BDBM50239167(CHEMBL1496110)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at mouse TRPC4 expressed in HEK293 cells coexpressing M5 receptor assessed as induction of TRPC4-mediated calcium influx by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50519475BDBM50519475(CHEMBL4438838)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77623BDBM77623(cid_46891894 | 4,6-dimethyl-2-(1-piperidinyl)quino...)
Affinity DataIC50: 5.49E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50519468BDBM50519468(CHEMBL4440241)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77626BDBM77626(cid_46891902 | 6-fluoro-4-methyl-2-(1-piperidinyl)...)
Affinity DataIC50: 6.18E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 85747BDBM85747(CLEMIZOLE HYDROCHLORIDE | NSC_2782 | CAS_442-52-4 ...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of YFP-tagged mouse TRPC4 beta expressed in thapsigargin treated HEK293 cells co-expressing M3 receptor assessed as reduction in carbachol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79618BDBM79618(N,N-diethyl-4-methyl-quinolin-2-amine;2,2,2-tris(f...)
Affinity DataIC50: 7.54E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 77622BDBM77622(4-methyl-2-(4-pyridin-4-ylpiperazin-1-yl)quinoline...)
Affinity DataIC50: 8.18E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50519472BDBM50519472(CHEMBL4454499)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of mouse TRPC4 expressed in HEK293 cells coexpressing M5 receptor assessed as reduction in TRPC4-mediated calcium influx by fluorescence m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79620BDBM79620(2-[4-(4-methyl-2-quinolinyl)-1-piperazinyl]benzoni...)
Affinity DataIC50: 8.90E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79622BDBM79622(1-(4-methylquinolin-2-yl)piperidin-3-ol;2,2,2-tris...)
Affinity DataIC50: 9.40E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79619BDBM79619(2-[4-(2-methoxyphenyl)piperazin-1-yl]-4-methylquin...)
Affinity DataIC50: 9.89E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79625BDBM79625(4,8-dimethyl-2-(1-pyrrolidinyl)quinoline;2,2,2-tri...)
Affinity DataIC50: 9.96E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273009BDBM50273009(CHEMBL4129809)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse TRPC4 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239166BDBM50239166(CHEMBL4083411)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at mouse TRPC4beta expressed in HEK293 cells co-expressing MOR decrease in DAMGO-evoked intracellular calcium level by Fluo-8-AM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492280BDBM50492280(CHEMBL2396911)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492279BDBM50492279(CHEMBL1376358)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492274BDBM50492274(CHEMBL2396912)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79617BDBM79617(2-(3,5-dimethylpiperidin-1-yl)-4-methyl-quinoline;...)
Affinity DataIC50: 1.19E+4nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50638821BDBM50638821(CHEMBL5561986)
Affinity DataIC50: 1.22E+4nMAssay Description:Antagonist activity at mouse TRPC4 stably expressed in HEK293 cells inhibition of calcium influx by calcium fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79621BDBM79621(VU0418913-1 | cid_46259350 | 4-(4-methyl-2-quinoli...)
Affinity DataIC50: 2.45E+4nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2011
Entry Details
PCBioAssay
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