Compile Data Set for Download or QSAR
Report error Found 186 of affinity data for UniProtKB/TrEMBL: Q9Y2T5
TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622923BDBM622923(US11780827, Example 21)
Affinity DataEC50:  2nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622939BDBM622939(US11780827, Example 37)
Affinity DataEC50:  3nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700723BDBM700723(US12115157, Ex. 13b)
Affinity DataEC50:  3nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622914BDBM622914(US11780827, Example 12)
Affinity DataEC50:  3nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622910BDBM622910(US11780827, Example 8)
Affinity DataEC50:  4nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622921BDBM622921(US11780827, Example 19)
Affinity DataEC50:  4nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622916BDBM622916(US11780827, Example 14)
Affinity DataEC50:  4nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622918BDBM622918(US11780827, Example 16)
Affinity DataEC50:  4nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622927BDBM622927(US11780827, Example 25)
Affinity DataEC50:  4nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622912BDBM622912(US11780827, Example 10)
Affinity DataEC50:  4nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622942BDBM622942(US11780827, Example 40)
Affinity DataEC50:  5nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622922BDBM622922(US11780827, Example 20)
Affinity DataEC50:  5nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622906BDBM622906(US11780827, Example 4)
Affinity DataEC50:  5nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622931BDBM622931(US11780827, Example 29)
Affinity DataEC50:  5nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622917BDBM622917(US11780827, Example 15)
Affinity DataEC50:  5nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50460255BDBM50460255(CHEMBL4226295)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622908BDBM622908(US11780827, Example 6)
Affinity DataEC50:  6nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622925BDBM622925(US11780827, Example 23)
Affinity DataEC50:  6nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622926BDBM622926(US11780827, Example 24)
Affinity DataEC50:  6nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622920BDBM622920(US11780827, Example 18)
Affinity DataEC50:  6nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622938BDBM622938(US11780827, Example 36)
Affinity DataEC50:  6nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622928BDBM622928(US11780827, Example 26)
Affinity DataEC50:  6nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622913BDBM622913(US11780827, Example 11)
Affinity DataEC50:  6nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700715BDBM700715(US12115157, Ex. 8b)
Affinity DataEC50:  7nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622924BDBM622924(US11780827, Example 22)
Affinity DataEC50:  7nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622948BDBM622948(US11780827, Example 46)
Affinity DataEC50:  7nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622937BDBM622937(US11780827, Example 35)
Affinity DataEC50:  8nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622932BDBM622932(US11780827, Example 30)
Affinity DataEC50:  8nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622934BDBM622934(US11780827, Example 32)
Affinity DataEC50:  8nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622940BDBM622940(US11780827, Example 38)
Affinity DataEC50:  9nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622903BDBM622903(US11780827, Example 1)
Affinity DataEC50:  9nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622904BDBM622904(US11780827, Example 2)
Affinity DataEC50:  9nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622915BDBM622915(US11780827, Example 13)
Affinity DataEC50:  9nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50460264BDBM50460264(CHEMBL4229128)
Affinity DataEC50:  9.60nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622907BDBM622907(US11780827, Example 5)
Affinity DataEC50:  10nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622909BDBM622909(US11780827, Example 7)
Affinity DataEC50:  10nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622935BDBM622935(US11780827, Example 33)
Affinity DataEC50:  10nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700720BDBM700720(US12115157, Ex. 11b)
Affinity DataEC50:  10nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622919BDBM622919(US11780827, Example 17)
Affinity DataEC50:  11nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700728BDBM700728(BDBM700731 | (S)—N-(3-cyano-4-fluorophenyl)-1,2,4-...)
Affinity DataEC50:  11nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700725BDBM700725(US12115157, Ex. 14b)
Affinity DataEC50:  11nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50252102BDBM50252102(CHEMBL4059658)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622929BDBM622929(US11780827, Example 27)
Affinity DataEC50:  11nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622941BDBM622941(US11780827, Example 39)
Affinity DataEC50:  12nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622943BDBM622943(US11780827, Example 41)
Affinity DataEC50:  12nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622930BDBM622930(US11780827, Example 28)
Affinity DataEC50:  12nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622947BDBM622947(US11780827, Example 45)
Affinity DataEC50:  14nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 622911BDBM622911(US11780827, Example 9)
Affinity DataEC50:  14nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2023
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700717BDBM700717(US12115157, Ex. 10a)
Affinity DataEC50:  14nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700707BDBM700707(US12115157, Ex. 1)
Affinity DataEC50:  15nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

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