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Found 375 with Last Name = 'sakaitani' and Initial = 'm'
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50002369((2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methyleth...)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50004899((1R,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50013055(2-aminopentanedioateglutamate | L-Glutamate | glut...)
Affinity DataKi:  118nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50013055(2-aminopentanedioateglutamate | L-Glutamate | glut...)
Affinity DataKi:  118nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50013055(2-aminopentanedioateglutamate | L-Glutamate | glut...)
Affinity DataKi:  131nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50002343(2-Methylamino-succinic acid | CHEMBL275325 | NMDA)
Affinity DataKi:  5.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50240399((2R,3R,4S)-3-(carboxymethyl)-4-isopropylpyrrolidin...)
Affinity DataKi:  6.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85210(DL-TBzOAsp)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85209(DL-THA)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85209(DL-THA)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85210(DL-TBzOAsp)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85211(t-2,4-PDC | t-PDC)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50240399((2R,3R,4S)-3-(carboxymethyl)-4-isopropylpyrrolidin...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50093753((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85210(DL-TBzOAsp)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85209(DL-THA)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50093753((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50240399((2R,3R,4S)-3-(carboxymethyl)-4-isopropylpyrrolidin...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85211(t-2,4-PDC | t-PDC)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM85211(t-2,4-PDC | t-PDC)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research

Curated by PDSP Ki Database
LigandPNGBDBM50093753((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50479835(CHEMBL510873)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479863(CHEMBL521743)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479859(CHEMBL508937)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479847(CHEMBL514300)
Affinity DataIC50:  1nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479856(CHEMBL454405)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479848(CHEMBL489318)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479849(CHEMBL489121)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479853(CHEMBL511113)
Affinity DataIC50:  2nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase(Candida albicans (Yeast))
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50096797(CHEMBL2370665 | macrocyclic lipopeptidolactone der...)
Affinity DataIC50:  2nMAssay Description:Inhibition of 1,3-beta-D-glucan synthase (GS) from candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50479850(CHEMBL475149)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479864(CHEMBL510021)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479860(CHEMBL473148)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
LigandPNGBDBM50479851(CHEMBL462021)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479857(CHEMBL472956)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479858(CHEMBL453395)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479836(CHEMBL511072)
Affinity DataIC50:  4nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase(Candida albicans (Yeast))
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50096795(CHEMBL2370654 | Macrocyclic lipopeptidolactone der...)
Affinity DataIC50:  5nMAssay Description:Inhibition of 1,3-beta-D-glucan synthase (GS) from candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50494481(CHEMBL3092178)
Affinity DataIC50:  5nMAssay Description:Inhibition of MEK1 (unknown origin) assessed as phosphorylation of Erk2 preincubated for 30 mins followed by FAM-Erktide addition measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase(Candida albicans (Yeast))
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50096793(CHEMBL2370666 | macrocyclic lipopeptidolactone der...)
Affinity DataIC50:  6nMAssay Description:Inhibition of 1,3-beta-D-glucan synthase (GS) from candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50479854(CHEMBL453394)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479837(CHEMBL516034)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50479838(CHEMBL513211)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50443366(CHEMBL3086065)
Affinity DataIC50:  7nMAssay Description:Inhibition of MEK1 (unknown origin) assessed as phosphorylation of Erk2 preincubated for 30 mins followed by FAM-Erktide addition measured after 60 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50479839(CHEMBL517280)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50494482(CHEMBL3092191)
Affinity DataIC50:  8nMAssay Description:Inhibition of C-Raf (unknown origin) assessed as phosphorylation of MEK1 after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase(Candida albicans (Yeast))
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50096799(CHEMBL2369134 | macrocyclic lipopeptidolactone der...)
Affinity DataIC50:  8nMAssay Description:Inhibition of 1,3-beta-D-glucan synthase (GS) from candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50443366(CHEMBL3086065)
Affinity DataIC50:  8nMAssay Description:Inhibition of C-Raf (unknown origin) assessed as phosphorylation of MEK1 after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50479861(CHEMBL473151)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM401184(8-Chloro-3-[(5-chloro-2-ethylsulfonylphenyl)methyl...)
Affinity DataIC50:  11nMAssay Description:DDR1 binding activity was measured using the LanthaScreen (Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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