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Found 136 with Last Name = 'tulinsky' and Initial = 'a'
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50076232((1S,7S)-7-Amino-7-benzyl-8-oxo-hexahydro-pyrazolo[...)
Affinity DataKi:  0.0710nMAssay Description:Binding affinity of the compound towards thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50228853((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  0.190nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50076233((3S,6R,8aR)-6-Amino-6-benzyl-5-oxo-octahydro-indol...)
Affinity DataKi:  0.650nMAssay Description:Binding affinity of the compound towards thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288457(CHEMBL317974 | macrocyclic tripeptide motif)
Affinity DataKi:  1nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50054502(CHEMBL140494 | N-((S)-3-Carbamimidoyl-2-hydroxy-cy...)
Affinity DataKi:  1.01nMAssay Description:compound was tested in vitro for inhibition of serine protease thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50052418((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288454(CHEMBL317527 | N-[3-((5S,20R,22aR)-5-Benzyl-4,7,18...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50076229((1S,7S)-7-Amino-7-benzyl-8-oxo-hexahydro-pyrazolo[...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity of the compound towards thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288451(CHEMBL319017 | N-{3-[(5S,15S,19R,21aR)-5-Benzyl-15...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50052417((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288453(CHEMBL317353 | N-[3-((5S,15S,19R,21aR)-5-Benzyl-4,...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50228853((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50052422((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50052418((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50052417((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50228863((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288457(CHEMBL317974 | macrocyclic tripeptide motif)
Affinity DataKi:  4.10nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50052422((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288453(CHEMBL317353 | N-[3-((5S,15S,19R,21aR)-5-Benzyl-4,...)
Affinity DataKi:  5.20nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288451(CHEMBL319017 | N-{3-[(5S,15S,19R,21aR)-5-Benzyl-15...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50228857((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  8.10nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50052425((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  8.20nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288454(CHEMBL317527 | N-[3-((5S,20R,22aR)-5-Benzyl-4,7,18...)
Affinity DataKi:  9.90nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataKi:  10nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50076230((3S,6S,8aR)-6-Amino-6-benzyl-5-oxo-octahydro-indol...)
Affinity DataKi:  10nMAssay Description:Binding affinity of the compound towards thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50228863((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  10nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288460(CHEMBL101049 | N-[3-((5S,18R,20aR)-5-Benzyl-4,7,16...)
Affinity DataKi:  10nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288458(CHEMBL431429 | N-[3-((5S,18R,20aR)-4,7,16,17,20-Pe...)
Affinity DataKi:  11nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50052423((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  12nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288459(CHEMBL317428 | N-[3-((5S,18R,20aR)-5-Benzyl-2-meth...)
Affinity DataKi:  13nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288452(CHEMBL99281 | N-[3-((5S,18R,20aR)-4,7,16,17,20-Pen...)
Affinity DataKi:  14nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288455(CHEMBL100712 | N-[3-((5S,21R,23aR)-5-Benzyl-4,7,19...)
Affinity DataKi:  15nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50052425((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  15nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288452(CHEMBL99281 | N-[3-((5S,18R,20aR)-4,7,16,17,20-Pen...)
Affinity DataKi:  20nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288460(CHEMBL101049 | N-[3-((5S,18R,20aR)-5-Benzyl-4,7,16...)
Affinity DataKi:  24nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288455(CHEMBL100712 | N-[3-((5S,21R,23aR)-5-Benzyl-4,7,19...)
Affinity DataKi:  25nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50052423((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  38nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50228856((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  50nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288450(CHEMBL328200 | N-[3-((6S,19R,21aR)-6-Benzyl-5,8,17...)
Affinity DataKi:  66nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50228855((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  73nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50228855((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  85nMAssay Description:Inhibition of human alpha-thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288450(CHEMBL328200 | N-[3-((6S,19R,21aR)-6-Benzyl-5,8,17...)
Affinity DataKi:  86nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288459(CHEMBL317428 | N-[3-((5S,18R,20aR)-5-Benzyl-2-meth...)
Affinity DataKi:  159nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288458(CHEMBL431429 | N-[3-((5S,18R,20aR)-4,7,16,17,20-Pe...)
Affinity DataKi:  163nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288456(CHEMBL430844 | N-[3-((5S,17R,19aR)-5-Benzyl-4,7,15...)
Affinity DataKi:  280nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50228857((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataKi:  290nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288461(CHEMBL98856 | N-[3-((5S,16R,18aR)-5-Benzyl-4,7,14,...)
Affinity DataKi:  473nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50288461(CHEMBL98856 | N-[3-((5S,16R,18aR)-5-Benzyl-4,7,14,...)
Affinity DataKi:  710nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM14111((2S)-N-[(2S)-1-(1-benzothiophen-2-yl)-5-carbamimid...)
Affinity DataKi:  1.34E+3nMAssay Description:Inhibition of bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50288456(CHEMBL430844 | N-[3-((5S,17R,19aR)-5-Benzyl-4,7,15...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
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