Compile Data Set for Download or QSAR
maximum 50k data
Found 39 with Last Name = 'almstead' and Initial = 'ji'
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474313(CHEMBL122698)
Affinity DataIC50:  510nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474311(Clinafloxacin)
Affinity DataIC50:  546nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474311(Clinafloxacin)
Affinity DataIC50:  2.73E+3nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474312(CHEMBL120948)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474318(CHEMBL123246)
Affinity DataIC50:  4.26E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474310(CHEMBL121176)
Affinity DataIC50:  4.61E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474316(CHEMBL331987)
Affinity DataIC50:  7.93E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474312(CHEMBL120948)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474315(CHEMBL421101)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221011(CHEMBL76485)
Affinity DataIC50:  8.61E+3nMAssay Description:Inhibitory activity against wild type gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474309(CHEMBL331076)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition effect on Escherichia coli Wild Type DNA gyrase Supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474317(CHEMBL122691)
Affinity DataIC50:  8.84E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)
Affinity DataIC50:  8.85E+3nMAssay Description:Inhibitory activity against wild type gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474316(CHEMBL331987)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474318(CHEMBL123246)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474319(CHEMBL420897)
Affinity DataIC50:  1.79E+4nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221010(CHEMBL79077)
Affinity DataIC50:  1.79E+4nMAssay Description:Inhibitory activity against wild type gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474313(CHEMBL122698)
Affinity DataIC50:  3.32E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474315(CHEMBL421101)
Affinity DataIC50:  3.37E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474317(CHEMBL122691)
Affinity DataIC50:  3.59E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)
Affinity DataIC50:  3.59E+4nMAssay Description:Inhibitory activity against quinolone resistant gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474319(CHEMBL420897)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474314(CHEMBL420884)
Affinity DataIC50:  6.94E+4nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474309(CHEMBL331076)
Affinity DataIC50:  7.15E+4nMAssay Description:Inhibition of Escherichia coli Quinolone resistant gyrase Supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221009(CHEMBL309434)
Affinity DataIC50:  9.02E+4nMAssay Description:Inhibitory activity against wild type gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221010(CHEMBL79077)
Affinity DataIC50:  1.06E+5nMAssay Description:Inhibitory activity against mammalian DNA topoisomerase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221010(CHEMBL79077)
Affinity DataIC50:  1.42E+5nMAssay Description:Inhibitory activity against quinolone resistant gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221008(CHEMBL80587)
Affinity DataIC50:  1.83E+5nMAssay Description:Inhibitory activity against wild type gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474314(CHEMBL420884)
Affinity DataIC50: >2.72E+5nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221011(CHEMBL76485)
Affinity DataIC50: >2.74E+5nMAssay Description:Inhibitory activity against quinolone resistant gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474310(CHEMBL121176)
Affinity DataIC50: >2.94E+5nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  3.07E+5nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221011(CHEMBL76485)
Affinity DataIC50:  4.03E+5nMAssay Description:Inhibitory activity against mammalian DNA topoisomerase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221009(CHEMBL309434)
Affinity DataIC50:  7.28E+5nMAssay Description:Inhibitory activity against mammalian DNA topoisomerase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221008(CHEMBL80587)
Affinity DataIC50: >1.45E+6nMAssay Description:Inhibitory activity against mammalian DNA topoisomerase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221008(CHEMBL80587)
Affinity DataIC50: >1.45E+6nMAssay Description:Inhibitory activity against quinolone resistant gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50221009(CHEMBL309434)
Affinity DataIC50: >1.45E+6nMAssay Description:Inhibitory activity against quinolone resistant gyrase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)
Affinity DataIC50: >1.66E+6nMAssay Description:Inhibitory activity against mammalian DNA topoisomerase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed