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Found 68 with Last Name = 'antonetti' and Initial = 'da'
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543625(CHEMBL3732444)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant full-length human aPKCzeta expressed in Sf21 insect cells using 5FAM-ERMRPRKRQGSVRRRV-NH2 as substrate in presence of ATP a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543619(CHEMBL4637651)
Affinity DataIC50:  70nMAssay Description:Inhibition of recombinant full-length human aPKCiota using CREBtide as substrate incubated for 3 hrs in presence of ATP by kinase Glo luminescent ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543624(CHEMBL3732675)
Affinity DataIC50:  270nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using ERMRPRKRQGSVRRRV as substrate in presence of ATP by ADP Quest kit assayMore data for this Ligand-Target Pair
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543617(CHEMBL4645321)
Affinity DataIC50:  360nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543616(CHEMBL4647507)
Affinity DataIC50:  380nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543614(CHEMBL4635556)
Affinity DataIC50:  420nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543619(CHEMBL4637651)
Affinity DataIC50:  520nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543618(CHEMBL4640268)
Affinity DataIC50:  560nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543621(CHEMBL4633210)
Affinity DataIC50:  700nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139465(US8889672, 317-080-001)
Affinity DataIC50:  800nMAssay Description:Inhibition of atypical PKCzeta (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139465(US8889672, 317-080-001)
Affinity DataIC50:  900nMAssay Description:Inhibition of atypical PKCiota (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139469(US8889672, 317-052-004)
Affinity DataIC50:  900nMAssay Description:Inhibition of atypical PKCiota (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139465(US8889672, 317-080-001)
Affinity DataIC50:  1.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Penn State University College Of Medicine

Curated by ChEMBL
LigandPNGBDBM139469(US8889672, 317-052-004)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543622(CHEMBL4649467)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543619(CHEMBL4637651)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of recombinant full-length human aPKCzeta in presence of ATP at Km concentration by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139466(US8889672, 317-094-001)
Affinity DataIC50:  2.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139467(US8889672, 268-020-002)
Affinity DataIC50:  2.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139469(US8889672, 317-052-004)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of atypical PKCzeta (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139467(US8889672, 268-020-002)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of atypical PKCiota (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139467(US8889672, 268-020-002)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of atypical PKCzeta (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139466(US8889672, 317-094-001)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of atypical PKCzeta (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543615(CHEMBL4648499)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139483(US8889672, 194-094-003)
Affinity DataIC50:  3.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543626(CHEMBL3729812)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant full-length human aPKCzeta expressed in Sf21 insect cells using 5FAM-ERMRPRKRQGSVRRRV-NH2 as substrate in presence of ATP a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139468(US8889672, 317-054-001)
Affinity DataIC50:  4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139480(US8889672, 194-074-005)
Affinity DataIC50:  4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139481(US8889672, 194-074-008)
Affinity DataIC50:  4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139468(US8889672, 317-054-001)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of atypical PKCzeta (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543619(CHEMBL4637651)
Affinity DataIC50:  4.08E+3nMAssay Description:Inhibition of recombinant full-length human aPKCiota in presence of ATP at Km concentration by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139482(US8889672, 194-094-008)
Affinity DataIC50:  5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139484(US8889672, 194-094-009)
Affinity DataIC50:  5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C iota type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of atypical PKCiota (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139469(US8889672, 317-052-004)
Affinity DataIC50:  5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50:  6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139470(US8889672, 317-056-002)
Affinity DataIC50:  6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139471(US8889672, 317-120-001)
Affinity DataIC50:  6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139472(US8889672, 252-036-001)
Affinity DataIC50:  6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of atypical PKCzeta (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139472(US8889672, 252-036-001)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of atypical PKCzeta (unknown origin) using CREBtide as substrate incubated for 1 hr measured every 2.5 mins by ADP Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139473(US8889672, 227-076-001)
Affinity DataIC50:  7.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139474(US8889672, 317-052-001)
Affinity DataIC50:  7.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Penn State University College Of Medicine

Curated by ChEMBL
LigandPNGBDBM139465(US8889672, 317-080-001)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Penn State University College Of Medicine

Curated by ChEMBL
LigandPNGBDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Penn State University College Of Medicine

Curated by ChEMBL
LigandPNGBDBM139467(US8889672, 268-020-002)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139475(US8889672, 268-044-002)
Affinity DataIC50:  1.10E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543620(CHEMBL4640910)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50543623(CHEMBL4638392)
Affinity DataIC50:  1.62E+4nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139478(US8889672, 317-048-002)
Affinity DataIC50:  1.70E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50:  2.00E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
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