Compile Data Set for Download or QSAR
maximum 50k data
Found 440 with Last Name = 'hadden' and Initial = 'mk'
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257185((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-5-guanidino-2-...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257186((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-azido...)
Affinity DataKi:  0.730nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataKi:  1.05nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  1.64nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240844((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-aceta...)
Affinity DataKi:  1.81nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257188((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-5-guanidino-2-...)
Affinity DataKi:  2.01nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50300041(7-(3-(dimethylamino)propoxy)-6-methoxy-2-(4-methyl...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to human recombinant G9a catalytic domain amino acid 913 to 1193 expressed in Escherichia coli BL21 (DE3) by isothermal titration ca...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257194((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-(7-aminoheptanam...)
Affinity DataKi:  2.99nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50353128(CHEMBL1231795)
Affinity DataKi:  3.70nMAssay Description:Competitive inhibition of G9a by fluorescence polarization assay in presence of fluorescein-labeled H3 peptideMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257192((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-7-amino-3-a...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257187((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino...)
Affinity DataKi:  4.87nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257192((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-7-amino-3-a...)
Affinity DataKi:  5.49nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257189((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataKi:  8.07nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257193((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataKi:  9.90nMAssay Description:Binding affinity to human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257193((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataKi:  10.4nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257191((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-7-amino-3-(...)
Affinity DataKi:  20.3nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240339((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-5-g...)
Affinity DataKi:  95nMAssay Description:Binding affinity to human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257197((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataKi:  105nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257190((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3-acetamido...)
Affinity DataKi:  136nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240339((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-5-g...)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase, H3 lysine-79 specific(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50396023(CHEMBL2169919)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant DOT1L using [3H]-SAM as substrate after 30 minsMore data for this Ligand-Target Pair
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50396022(CHEMBL2169920)
Affinity DataKi:  300nMAssay Description:Competitive binding affinity to full length human SMYD2 amino acid 1 to 433 expressed in Escherichia coli BL21 (DE3) after 90 mins by radioactive fil...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257195((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataKi:  303nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50396014(CHEMBL2169888)
Affinity DataKi:  610nMAssay Description:Inhibition of LSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257199((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-(5-guani...)
Affinity DataKi:  631nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257196((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-2-acetamido...)
Affinity DataKi:  647nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50396015(CHEMBL2169921)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human LSD1 using histone H3 peptide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463119(CHEMBL4240676)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257198((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataKi:  2.17E+3nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50346874(CHEMBL1797649)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of recombinant LSD1 catalytic domain amino acid 178 to 831 expressed in Sf9 cells infected with baculovirus using diMeK4H3-21 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463115(CHEMBL1717725)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50346862(CHEMBL1215658)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of N terminal hexahistidine-tag recombinant human LSD1 expressed in Escherichia coli BL21 (DE3) using histone H3 peptide as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463120(CHEMBL1721787)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463107(CHEMBL4245882)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463117(CHEMBL4249624)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463116(CHEMBL4237457)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463122(CHEMBL4249812)
Affinity DataKi:  4.80E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463118(CHEMBL4246571)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50346534(CHEMBL1797705)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of N terminal hexahistidine-tag recombinant human LSD1 expressed in Escherichia coli BL21 (DE3) using histone H3 peptide as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463106(CHEMBL4238011)
Affinity DataKi:  6.90E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463105(CHEMBL4244254)
Affinity DataKi:  7.40E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50346865(2-PFPA | CHEMBL1797642)
Affinity DataKi:  8.90E+3nMAssay Description:Inhibition of LSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463108(CHEMBL4244874)
Affinity DataKi:  8.90E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463113(CHEMBL4238016)
Affinity DataKi:  1.16E+4nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463114(CHEMBL4241371)
Affinity DataKi:  1.19E+4nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463103(CHEMBL4237396)
Affinity DataKi:  1.45E+4nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463123(CHEMBL4239688)
Affinity DataKi:  1.48E+4nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463111(CHEMBL4239342)
Affinity DataKi:  1.57E+4nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463109(CHEMBL4241418)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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