TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:TP_TRANSPORTER: transepithelial transport of digoxin (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 350nMAssay Description:TP_TRANSPORTER: transepithelial transport of digoxin (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 430nMAssay Description:TP_TRANSPORTER: transepithelial transport of digoxin (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 440nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 880nMAssay Description:TP_TRANSPORTER: transepithelial transport of digoxin (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 2.18E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 2.31E+3nMAssay Description:TP_TRANSPORTER: transepithelial transport of digoxin (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 8.11E+3nMAssay Description:TP_TRANSPORTER: inhibition of Vinblastine transepithelial transport (basal to apical) in MRP2-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 8.59E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(C.H.O.)
National Children'S Medical Research Center
Curated by PDSP Ki Database
National Children'S Medical Research Center
Curated by PDSP Ki Database
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 1.15E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:TP_TRANSPORTER: transepithelial transport of digoxin (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 1.51E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 2.64E+4nMAssay Description:TP_TRANSPORTER: inhibition of Vinblastine transepithelial transport (basal to apical) in MRP2-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 4.94E+4nMAssay Description:TP_TRANSPORTER: inhibition of Vinblastine transepithelial transport (basal to apical) in MRP2-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 1.11E+5nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 1.40E+5nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 2.13E+5nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 2.95E+5nMAssay Description:TP_TRANSPORTER: inhibition of Vinblastine transepithelial transport (basal to apical) in MRP2-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 7.56E+5nMAssay Description:TP_TRANSPORTER: inhibition of Vinblastine transepithelial transport (basal to apical) in MRP2-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 7.68E+5nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) in MDR1-expressing MDCK cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
The University Of Kansas
Curated by ChEMBL
The University Of Kansas
Curated by ChEMBL
Affinity DataKi: 8.02E+5nMAssay Description:TP_TRANSPORTER: inhibition of Vinblastine transepithelial transport (basal to apical) in MRP2-expressing MDCK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibitory concentration against Selectin E expressed at the inflammatory lesion was measured by inhibition of leukocyte rolling in the inflammatory ...More data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences
Curated by ChEMBL
National Institute Of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 0.0100nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences
Curated by ChEMBL
National Institute Of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 0.680nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences
Curated by ChEMBL
National Institute Of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 0.210nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences
Curated by ChEMBL
National Institute Of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 0.0440nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences
Curated by ChEMBL
National Institute Of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 0.150nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences
Curated by ChEMBL
National Institute Of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 0.290nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair