Affinity DataKi: 0.994nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.994nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.43nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.53nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 25.6nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 42.9nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 129nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 129nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 273nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 373nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 422nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 441nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 441nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 445nMAssay Description:Binding affinity towards mu Opioid receptor in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 849nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.76E+3nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.22E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 3.04E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.57E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.57E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 4.17E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 4.83E+3nMAssay Description:Binding affinity towards mu Opioid receptor in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.99E+3nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 5.06E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 8.16E+3nMAssay Description:Evaluated for its ability to displace [3H]DAGO binding to Opioid receptor mu 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 8.16E+3nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.81E+4nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: >3.80E+5nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibitory activity towards delta Opioid receptor using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibitory activity towards Opioid receptor mu 1 using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 246nMAssay Description:Inhibitory activity towards Opioid receptor mu 1 using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
Affinity DataIC50: 279nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair