Affinity DataKi: 1.30E+3nM ΔG°: -34.9kJ/mole IC50: 800nMpH: 7.5 T: 2°CAssay Description:Briefly, Bc-SMase (50 ng/ml) was treated at 37 °C for 60 min with various compounds that were solubilized in dimethylacetoamide. The reaction mix...More data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nM ΔG°: -33.0kJ/mole IC50: 900nMpH: 7.5 T: 2°CAssay Description:Briefly, Bc-SMase (50 ng/ml) was treated at 37 °C for 60 min with various compounds that were solubilized in dimethylacetoamide. The reaction mix...More data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nM ΔG°: -31.4kJ/mole IC50: 1.20E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, Bc-SMase (50 ng/ml) was treated at 37 °C for 60 min with various compounds that were solubilized in dimethylacetoamide. The reaction mix...More data for this Ligand-Target Pair
Affinity DataIC50: 0.720nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 1 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 1 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 169nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 1 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 1 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 772nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 908nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 995nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 1 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 1 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair