Compile Data Set for Download or QSAR
maximum 50k data
Found 52 with Last Name = 'winkler' and Initial = 'da'
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50423836(CHEMBL1829034)
Affinity DataIC50:  0.0700nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50105400((S)-2-{[(S)-2-(3,4-Dimethoxy-benzenesulfonyl)-1,2,...)
Affinity DataIC50:  0.530nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50095248((S)-2-[((S)-1-Benzyl-5-oxo-pyrrolidine-2-carbonyl)...)
Affinity DataIC50:  0.540nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50423837(CHEMBL1829035)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50124286(3-(2'-Methoxy-biphenyl-4-yl)-2-{[1-((S)-toluene-4-...)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50423833(CHEMBL1828842)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50423830(CHEMBL1828839)
Affinity DataIC50:  4.5nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50423832(CHEMBL1828841)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50117056((S)-2-(2-Bromo-6-methyl-benzoylamino)-3-[4-(2,6-di...)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50113545((S)-2-[(4,5-Dihydro-pyrazole-1-carbonyl)-amino]-3-...)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50119087((S)-2-(2-Chloro-benzoylamino)-3-(2'-{[2-(4-hydroxy...)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50116198((S)-2-[2-(2-Chloro-phenyl)-acetylamino]-3-(2'-meth...)
Affinity DataIC50:  37nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50089009((S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amin...)
Affinity DataIC50:  60nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50423835(CHEMBL1829033)
Affinity DataIC50:  67nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50423834(CHEMBL1829032)
Affinity DataIC50:  105nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50144767((S)-2-{[(S)-1-(3,5-Dichloro-benzenesulfonyl)-pyrro...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50117076((S)-3-[4-(2,6-Dichloro-benzoylamino)-phenyl]-2-[(2...)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2C1(Rattus norvegicus)
Csiro Division Of Chemicals And Polymers

Curated by ChEMBL
LigandPNGBDBM50367914(CHEMBL1794796)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against Mannosidase in jack bean (Canavalia ensiformis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2C1(Rattus norvegicus)
Csiro Division Of Chemicals And Polymers

Curated by ChEMBL
LigandPNGBDBM50367915(CHEMBL1794797)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against Mannosidase in jack bean (Canavalia ensiformis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | CHEM...)
Affinity DataIC50:  900nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAlpha-mannosidase 2C1(Rattus norvegicus)
Csiro Division Of Chemicals And Polymers

Curated by ChEMBL
LigandPNGBDBM50016706(CHEMBL63139 | Octahydro-indolizine-1,2,8-triol | S...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibitory activity against Mannosidase in jack bean (Canavalia ensiformis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50087592((S)-3-(4-Pentyloxy-phenyl)-2-[(pyridine-3-carbonyl...)
Affinity DataIC50:  3.80E+3nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50114294((S)-3-[4-(2,6-Dichloro-benzoylamino)-phenyl]-2-(4,...)
Affinity DataIC50:  4.00E+3nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Ian Wark Laboratories

Curated by ChEMBL
LigandPNGBDBM50423831(CHEMBL1828840)
Affinity DataIC50:  4.10E+3nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCadherin-2(Homo sapiens (Human))
Csiro Materials Science And Engineering

Curated by ChEMBL
LigandPNGBDBM50339160(CHEMBL1689350 | N-Ac-CHAVDC-NH2)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at N-cadherinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326770(4-isobutyl-5-methylene-2-oxo-1-(2,4,5-trichlorophe...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326767(4-butyl-1-(2-tert-butyl-5-chlorophenyl)-5-methylen...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326755(1-(2,5-di-tert-butylphenyl)-4-methyl-5-methylene-2...)
Affinity DataIC50:  6.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326760(4-ethyl-5-methylene-2-oxo-1-(2,4,5-trichlorophenyl...)
Affinity DataIC50:  7.25E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326765(4-butyl-1-(3-chloro-2-methylphenyl)-5-methylene-2-...)
Affinity DataIC50:  8.30E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326758(1-(4-tert-butyl-2,5-dichlorophenyl)-4-methyl-5-met...)
Affinity DataIC50:  8.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326759(1-(2-tert-butyl-5-chlorophenyl)-4-ethyl-5-methylen...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326766(4-butyl-1-(5-chloro-2-methylphenyl)-5-methylene-2-...)
Affinity DataIC50:  1.25E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326773(1-cyclohexyl-5-methylene-2-oxo-4-phenyl-2,5-dihydr...)
Affinity DataIC50:  1.25E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326761(1-(2-tert-butylphenyl)-4-isopropyl-5-methylene-2-o...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326774(3-benzoyl-4-methyl-5-methylene-1-(3-(trifluorometh...)
Affinity DataIC50:  1.75E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326756(1-(2,6-diisopropylphenyl)-4-methyl-5-methylene-2-o...)
Affinity DataIC50:  2.35E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326757(1-(3,5-dichlorophenyl)-4-methyl-5-methylene-2-oxo-...)
Affinity DataIC50:  2.75E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326769(4-butyl-1-(2-ethyl-6-methylphenyl)-5-methylene-2-o...)
Affinity DataIC50:  3.30E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326762(1-(2-tert-butyl-4-chlorophenyl)-4-isopropyl-5-meth...)
Affinity DataIC50:  4.20E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326763(4-isopropyl-1-(2-isopropyl-6-methylphenyl)-5-methy...)
Affinity DataIC50:  4.70E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326754(4-methyl-5-methylene-2-oxo-1-(2-(trifluoromethyl)p...)
Affinity DataIC50:  4.80E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326772(1-(2-isopropyl-6-methylphenyl)-5-methylene-2-oxo-4...)
Affinity DataIC50:  5.50E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326768(4-butyl-1-(2-chloro-6-methylphenyl)-5-methylene-2-...)
Affinity DataIC50:  5.60E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2C1(Rattus norvegicus)
Csiro Division Of Chemicals And Polymers

Curated by ChEMBL
LigandPNGBDBM50016703(2-Hydroxymethyl-pyrrolidine-3,4-diol | BDBM5003148...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibitory activity against Mannosidase in jack bean (Canavalia ensiformis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2C1(Rattus norvegicus)
Csiro Division Of Chemicals And Polymers

Curated by ChEMBL
LigandPNGBDBM50403114(CHEMBL1337303)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibitory activity against Mannosidase in jack bean (Canavalia ensiformis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326771(4-isobutyl-1-mesityl-5-methylene-2-oxo-2,5-dihydro...)
Affinity DataIC50:  1.75E+5nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326775(CHEMBL1254537 | N,1-Bis(3-chlorophenyl)-4-methyl-5...)
Affinity DataIC50:  2.50E+5nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326764(1-(2,4-dichloro-6-methylphenyl)-4-isopropyl-5-meth...)
Affinity DataIC50:  4.80E+5nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 52 total ) | Next | Last >>
Jump to: