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Found 6 Enz. Inhib. hit(s) with all data for entry = 2474
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM367610(N-[(1S)-2-[4-[2- (4-Amino-2- chloro-6-methyl- pyri...)
Affinity DataIC50:  54.4nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM367613(N-[(1S)-2-[4-[2-(4-Amino-6-chloro-2-methyl-pyrimid...)
Affinity DataIC50:  68.9nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM367612(N-[(1S)-2-[4-[2-(4-Amino-6-chloro-2-methyl-pyrimid...)
Affinity DataIC50:  96.4nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM367615(Methyl N-[(1S)-2-[4-[2-(4-amino-6-chloro-2-methyl-...)
Affinity DataIC50:  149nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM367614(N-[(1S)-2-[4-[2-(4-Amino-6-chloro-2-methyl-pyrimid...)
Affinity DataIC50:  170nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM367611(N-[(1S)-2-[(4R,S)- 4-[2-(4-Amino-6- chloro-2-methy...)
Affinity DataIC50:  574nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent