Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 5865
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM97725(US8476267, 2)
Affinity DataIC50:  22nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM50390707(CHEMBL2070316 | US8486964, 1)
Affinity DataIC50:  26nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM50390706(CHEMBL2070315 | US8486964, 4)
Affinity DataIC50:  46nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Merck Patent

US Patent
LigandPNGBDBM50390706(CHEMBL2070315 | US8486964, 4)
Affinity DataIC50:  490nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck Patent

US Patent
LigandPNGBDBM50390707(CHEMBL2070316 | US8486964, 1)
Affinity DataIC50:  670nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck Patent

US Patent
LigandPNGBDBM50390706(CHEMBL2070315 | US8486964, 4)
Affinity DataIC50:  780nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Merck Patent

US Patent
LigandPNGBDBM50390707(CHEMBL2070316 | US8486964, 1)
Affinity DataIC50:  930nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Merck Patent

US Patent
LigandPNGBDBM97725(US8476267, 2)
Affinity DataIC50:  1.29E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck Patent

US Patent
LigandPNGBDBM97725(US8476267, 2)
Affinity DataIC50:  1.54E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of 11-beta-HSD-1 enzyme assay using human recombinant 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-HSD-1) enzyme was expressed in ...More data for this Ligand-Target Pair
In DepthDetails US Patent