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Found 29 Enz. Inhib. hit(s) with all data for entry = 6568
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139465(US8889672, 317-080-001)
Affinity DataIC50:  1.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139466(US8889672, 317-094-001)
Affinity DataIC50:  2.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139467(US8889672, 268-020-002)
Affinity DataIC50:  2.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139483(US8889672, 194-094-003)
Affinity DataIC50:  3.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139468(US8889672, 317-054-001)
Affinity DataIC50:  4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139481(US8889672, 194-074-008)
Affinity DataIC50:  4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139480(US8889672, 194-074-005)
Affinity DataIC50:  4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139469(US8889672, 317-052-004)
Affinity DataIC50:  5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139482(US8889672, 194-094-008)
Affinity DataIC50:  5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139484(US8889672, 194-094-009)
Affinity DataIC50:  5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139470(US8889672, 317-056-002)
Affinity DataIC50:  6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50:  6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139472(US8889672, 252-036-001)
Affinity DataIC50:  6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139471(US8889672, 317-120-001)
Affinity DataIC50:  6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139474(US8889672, 317-052-001)
Affinity DataIC50:  7.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139473(US8889672, 227-076-001)
Affinity DataIC50:  7.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139475(US8889672, 268-044-002)
Affinity DataIC50:  1.10E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139478(US8889672, 317-048-002)
Affinity DataIC50:  1.70E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139477(US8889672, 317-008-004)
Affinity DataIC50:  2.00E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50:  2.00E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139476(US8889672, 317-010-004)
Affinity DataIC50:  2.10E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139488(US8889672, 5627112 | US8889672, 5632675)
Affinity DataIC50:  2.40E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139486(US8889672, 5132573)
Affinity DataIC50:  2.60E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139488(US8889672, 5627112 | US8889672, 5632675)
Affinity DataIC50:  2.80E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50:  3.50E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139489(US8889672, APOGEE A)
Affinity DataIC50:  3.90E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139487(US8889672, 5311310)
Affinity DataIC50:  4.10E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139491(US8889672, 5635527)
Affinity DataIC50:  6.20E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM139492(US8889672, APOGEE B)
Affinity DataIC50:  7.10E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent