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Found 13 Enz. Inhib. hit(s) with all data for entry = 50017282
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180049(3-[2-isobutoxy-5-(4-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180047(3-[2-isobutoxy-5-(3-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180051((R)-4-(4-methylpentanoyl)-8-(4-methylpentylidene)-...)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180048((R)-8-(3-methylbutylidene)-4-(5-methylhexanoyl)-1-...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180050(3-[2-benzyloxy-5-(4-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  4.20E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180048((R)-8-(3-methylbutylidene)-4-(5-methylhexanoyl)-1-...)
Affinity DataIC50:  4.60E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180047(3-[2-isobutoxy-5-(3-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  6.00E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180049(3-[2-isobutoxy-5-(4-isobutoxybenzoyl)phenyl]propio...)
Affinity DataIC50:  6.10E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180051((R)-4-(4-methylpentanoyl)-8-(4-methylpentylidene)-...)
Affinity DataIC50:  6.50E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180052(3-[5-(4-isobutoxybenzoyl)-2-propoxyphenyl]propioni...)
Affinity DataIC50:  9.10E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180046(3-[2-isobutoxy-5-(4-propoxybenzoyl)phenyl]propioni...)
Affinity DataIC50:  9.30E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180053(3-(5-benzoyl-2-isobutoxyphenyl)propionic acid | CH...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50180045(3-[3-(4-isobutoxybenzoyl)phenyl]propionic acid | C...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed