Found 30 Enz. Inhib. hit(s) with all data for entry = 50040089 TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 1.86nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 4.57nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 5.01nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 7.76nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 9.12nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 11.0nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 12.3nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 15.5nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 23.4nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 26.3nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 50.1nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Antagonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as inhibition of increase in intracellular calcium compound pr...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 8.91E+3nMAssay Description:Antagonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as inhibition of increase in intracellular calcium compound pr...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 2.63E+4nMAssay Description:Partial agonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as increase in intracellular calcium using Fluo-R stainin...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Agonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as increase in intracellular calcium using Fluo-R staining by mic...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Agonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as increase in intracellular calcium using Fluo-R staining by mic...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 81.3nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 148nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 35.5nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 224nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 66.1nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 25.1nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 708nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 339nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 676nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 195nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 661nMAssay Description:Partial agonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as increase in intracellular calcium using Fluo-R stainin...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
