Compile Data Set for Download or QSAR
maximum 50k data
Found 56 Enz. Inhib. hit(s) with all data for entry = 50039802
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384423(CHEMBL2031485 | US9896452, Example 62)
Affinity DataIC50:  0.800nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384412(CHEMBL2031504)
Affinity DataIC50:  0.800nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384437(CHEMBL2031501)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384436(CHEMBL2031500)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384417(CHEMBL2031478)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384408(CHEMBL2031498)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384428(CHEMBL2031491 | US9896452, Example 8)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384429(CHEMBL2031492 | US9896452, Example 137)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384408(CHEMBL2031498)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384417(CHEMBL2031478)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384419(CHEMBL2031480)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384419(CHEMBL2031480)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384418(CHEMBL2031479)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384415(CHEMBL2031507)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384420(CHEMBL2031482)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384430(CHEMBL2031493 | US9896452, Example 12)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384411(CHEMBL2031503)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384411(CHEMBL2031503)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384426(CHEMBL2031489 | US9896452, Example 9)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384420(CHEMBL2031482)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384421(CHEMBL2031483)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384412(CHEMBL2031504)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384422(CHEMBL2031484 | US9896452, Example 125)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384423(CHEMBL2031485 | US9896452, Example 62)
Affinity DataIC50:  8.70nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384409(CHEMBL2031487 | US9896452, Example 138)
Affinity DataIC50:  9nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384427(CHEMBL2031490 | US9896452, Example 139)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384413(CHEMBL2031505)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384436(CHEMBL2031500)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384421(CHEMBL2031483)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384414(CHEMBL2031506)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384424(CHEMBL2031486 | US9896452, Example 124)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384418(CHEMBL2031479)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384435(CHEMBL2031499)
Affinity DataIC50:  27nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384427(CHEMBL2031490 | US9896452, Example 139)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384431(CHEMBL2031494)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384416(CHEMBL2111553 | CHEMBL291536 | SB-334867)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384409(CHEMBL2031487 | US9896452, Example 138)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384426(CHEMBL2031489 | US9896452, Example 9)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384428(CHEMBL2031491 | US9896452, Example 8)
Affinity DataIC50:  58nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384431(CHEMBL2031494)
Affinity DataIC50:  62nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384429(CHEMBL2031492 | US9896452, Example 137)
Affinity DataIC50:  82nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384414(CHEMBL2031506)
Affinity DataIC50:  96nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384410(CHEMBL2031502)
Affinity DataIC50:  121nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384415(CHEMBL2031507)
Affinity DataIC50:  125nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384435(CHEMBL2031499)
Affinity DataIC50:  137nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384425(CHEMBL2031488)
Affinity DataIC50:  145nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384432(CHEMBL2031495)
Affinity DataIC50:  146nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384413(CHEMBL2031505)
Affinity DataIC50:  151nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384424(CHEMBL2031486 | US9896452, Example 124)
Affinity DataIC50:  221nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50384434(CHEMBL2031497)
Affinity DataIC50:  390nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 56 total ) | Next | Last >>
Jump to: