Found 50 Enz. Inhib. hit(s) with all data for entry = 50036238 
Affinity DataKi: 1.30nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Affinity for A1 Adenosine receptor in rat brain using [3H]CHAMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 167nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 184nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 267nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 656nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 657nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.52E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 167nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 153nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 475nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 8.20nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 6.05E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 730nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 84nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.43E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.37E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
Affinity DataEC50: 332nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
