Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50036669
LigandPNGBDBM50067566((S)-2-{[2'-Ethyl-5-(pyridin-3-yloxymethyl)-bipheny...)
Affinity DataIC50:  0.350nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067563((S)-2-{[2'-Methyl-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067581((S)-2-{[2'-Methyl-5-(pyridin-3-ylaminomethyl)-biph...)
Affinity DataIC50:  0.420nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067559((S)-4-Methylsulfanyl-2-{[5-(pyridin-3-yloxymethyl)...)
Affinity DataIC50:  0.5nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  0.5nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067569((S)-2-{[2'-Chloro-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50:  0.610nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067568((S)-2-{[2'-Methyl-5-(pyridin-3-ylsulfanylmethyl)-b...)
Affinity DataIC50:  0.690nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067574((S)-2-({2'-Methyl-5-[(pyridin-3-ylmethyl)-amino]-b...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067557((S)-2-({2'-Methyl-5-[(pyridine-3-carbonyl)-amino]-...)
Affinity DataIC50:  1.60nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067564((S)-2-{[2'-Methoxy-5-(pyridin-3-yloxymethyl)-biphe...)
Affinity DataIC50:  3.30nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067565((S)-4-Methylsulfanyl-2-{[5-(pyridin-3-yloxymethyl)...)
Affinity DataIC50:  4.30nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067562((S)-2-{[3'-Methyl-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50:  5.40nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067572((S)-4-Methylsulfanyl-2-{[5-(pyridin-3-ylmethoxy)-b...)
Affinity DataIC50:  6.60nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067578((S)-4-Methylsulfanyl-2-{[5-(pyridin-3-ylaminomethy...)
Affinity DataIC50:  6.80nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067560((S)-4-Methylsulfanyl-2-{[5-(pyridin-3-ylsulfanylme...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067582((S)-2-{[3'-Methoxy-5-(pyridin-3-yloxymethyl)-biphe...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067561((S)-4-Methanesulfonyl-2-{[5-(pyridin-3-ylaminometh...)
Affinity DataIC50:  17nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067558((S)-4-Methylsulfanyl-2-({5-[(pyridin-3-ylmethyl)-a...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067583((S)-4-Carbamoyl-2-{[5-(pyridin-3-yloxymethyl)-biph...)
Affinity DataIC50:  48nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067571((S)-4-Methylsulfanyl-2-({5-[(pyridine-3-carbonyl)-...)
Affinity DataIC50:  70nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067570((R)-4-Methylsulfanyl-2-{[5-(pyridin-3-ylaminomethy...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067585((S)-2-{Methyl-[5-(pyridin-3-ylaminomethyl)-bipheny...)
Affinity DataIC50:  160nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067586((S)-2-{[4'-Methoxy-5-(pyridin-3-yloxymethyl)-biphe...)
Affinity DataIC50:  230nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067567((S)-2-{[4'-Methyl-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50:  360nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067576((S)-4-Methylsulfanyl-2-{[5-(pyridine-3-sulfonylmet...)
Affinity DataIC50:  550nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067577((S)-4-Methylsulfanyl-2-({5-[(pyridine-2-carbonyl)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067580((R)-3-Methylsulfanyl-2-{[5-(pyridin-3-yloxymethyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067579((S)-4-Methoxy-2-{[5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067575((S)-4-Methylsulfanyl-2-({5-[(pyridine-4-carbonyl)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067573((S)-2-{[5-(Pyridin-3-yloxymethyl)-biphenyl-2-carbo...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of farnesyltransferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed