Compile Data Set for Download or QSAR
maximum 50k data
Found 95 of affinity data for UniProtKB/TrEMBL: Q01177
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50074920(((R)-3-Phenyl-1-{(S)-2-phenyl-1-[3,3,3-trifluoro-1...)
Affinity DataKi:  40nMAssay Description:Inhibitory activity of compound against Plasmin (HP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50074921([(R)-1-({(S)-Naphthalen-2-yl-[3,3,3-trifluoro-1-(4...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity of compound against Plasmin (HP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50074915(((R)-2-Methyl-1-{(S)-2-phenyl-1-[3,3,3-trifluoro-1...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity of compound against Plasmin (HP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50074918(((R)-2,2-Dimethyl-1-{(S)-2-phenyl-1-[3,3,3-trifluo...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity of compound against Plasmin (HP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98600((2S)-2-[[(2R)-2-(benzylsulfonylamino)-3-hydroxy-pr...)
Affinity DataKi:  200nM ΔG°:  -38.1kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98587((2R)-N-[(1S)-1-(benzyloxymethyl)-2-[(4-carbamimido...)
Affinity DataKi:  270nM ΔG°:  -37.4kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98599((2S)-6-amino-2-[[(2R)-2-(benzylsulfonylamino)-3-hy...)
Affinity DataKi:  360nM ΔG°:  -36.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98603(3-amino-N-[4-[[(2S)-2-[[(2R)-2-(benzylsulfonylamin...)
Affinity DataKi:  400nM ΔG°:  -36.4kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50074916([(R)-2,2-Dimethyl-1-({(S)-naphthalen-2-yl-[3,3,3-t...)
Affinity DataKi:  500nMAssay Description:Inhibitory activity of compound against Plasmin (HP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98601((2S)-6-[[2-[2-[2-[2-[2-[2-[2-[2-[2-(2-aminoethoxy)...)
Affinity DataKi:  530nM ΔG°:  -35.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50074917(Morpholine-4-carboxylic acid ((R)-2,2-dimethyl-1-{...)
Affinity DataKi:  560nMAssay Description:Inhibitory activity of compound against Plasmin (HP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50076221((S)-1-((R)-2-Amino-3-phenyl-propionyl)-pyrrolidine...)
Affinity DataKi:  699nMAssay Description:Inhibitory concentration of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50231520((R)-N-[(S)-1-(4-carbamimidoyl-benzylcarbamoyl)-2-h...)
Affinity DataKi:  750nM ΔG°:  -34.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98588((2S)-3-amino-2-[[(2R)-2-(benzylsulfonylamino)-3-hy...)
Affinity DataKi:  810nM ΔG°:  -34.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98593(US8476306, 6.19 | methyl 4-[[(1R)-2-[[(1S)-2-[(4-c...)
Affinity DataKi:  960nM ΔG°:  -34.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50076220((1S,7S)-7-Amino-7-benzyl-hexahydro-pyrazolo[1,2-a]...)
Affinity DataKi:  978nMAssay Description:Inhibitory concentration of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98590((2S)-3-benzyloxy-2-[[(2R)-2-(benzylsulfonylamino)-...)
Affinity DataKi:  1.10E+3nM ΔG°:  -33.9kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98589((2S)-2-[[(2R)-2-(benzylsulfonylamino)-3-hydroxy-pr...)
Affinity DataKi:  1.40E+3nM ΔG°:  -33.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98583(4-[[(1R)-2-[[(1S)-2-[(4-carbamimidoylphenyl)methyl...)
Affinity DataKi:  3.00E+3nM ΔG°:  -31.4kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98591(3-[[(1R)-2-[[(1S)-2-[(4-carbamimidoylphenyl)methyl...)
Affinity DataKi:  4.20E+3nM ΔG°:  -30.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98584(3-[[(1R)-2-[[(1S)-2-[(4-carbamimidoylphenyl)methyl...)
Affinity DataKi:  4.70E+3nM ΔG°:  -30.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50147046(5-Methylsulfanyl-4-[4-(5-propoxy-1-pyridin-2-yl-1H...)
Affinity DataKi:  5.00E+3nMAssay Description:In vitro binding affinity towards plasmin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98592(4-[[(1R)-2-[[(1S)-2-[(4-carbamimidoylphenyl)methyl...)
Affinity DataKi:  6.20E+3nM ΔG°:  -29.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98586((2R)-2-[[4-(aminomethyl)phenyl]methylsulfonylamino...)
Affinity DataKi:  7.40E+3nM ΔG°:  -29.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98602(3-amino-N-[4-[[2-[[(2R)-3-amino-2-(benzylsulfonyla...)
Affinity DataKi:  9.60E+3nM ΔG°:  -28.5kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50110015(CHEMBL158936 | N-(BENZYLSULFONYL)SERYL-N~1~-{4-[AM...)
Affinity DataKi:  1.10E+4nM ΔG°:  -28.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98579(US8476306, 6.4 | methyl 4-[[(1R)-2-[[2-[(4-carbami...)
Affinity DataKi:  1.70E+4nM ΔG°:  -27.1kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98595((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  1.80E+4nM ΔG°:  -27.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98596((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  2.00E+4nM ΔG°:  -26.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50069190(CHEMBL287614 | N-(1-Carbamimidoyl-piperidin-4-ylme...)
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity against serine protease plasminMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98604(2-[4-[[(1R)-2-[[2-[4-[(3-amino-4-methoxy-benzoyl)a...)
Affinity DataKi:  2.70E+4nM ΔG°:  -26.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98585((2R)-N-[(1S)-2-[(4-carbamimidoylphenyl)methylamino...)
Affinity DataKi:  2.70E+4nM ΔG°:  -26.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50110015(CHEMBL158936 | N-(BENZYLSULFONYL)SERYL-N~1~-{4-[AM...)
Affinity DataKi:  2.80E+4nM ΔG°:  -25.9kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98597((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  3.20E+4nM ΔG°:  -25.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98594((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  3.20E+4nM ΔG°:  -25.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98580(4-[[(1R)-2-[[2-[(4-carbamimidoylphenyl)methylamino...)
Affinity DataKi:  3.50E+4nM ΔG°:  -25.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98598((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  3.70E+4nM ΔG°:  -25.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98581(US8476306, 6.6 | methyl 2-[[(1R)-2-[[2-[(4-carbami...)
Affinity DataKi:  3.80E+4nM ΔG°:  -25.1kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98578(3-[[(1R)-2-[[2-[(4-carbamimidoylphenyl)methylamino...)
Affinity DataKi:  5.90E+4nM ΔG°:  -24.1kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50074919(Morpholine-4-carboxylic acid [(R)-2,2-dimethyl-1-(...)
Affinity DataKi:  1.10E+5nMAssay Description:Inhibitory activity of compound against Plasmin (HP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50368379(CHEMBL1202120)
Affinity DataKi:  1.57E+5nMAssay Description:In vitro inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM98582(2-[[(1R)-2-[[2-[(4-carbamimidoylphenyl)methylamino...)
Affinity DataKi:  2.20E+5nM ΔG°:  -20.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against PlasminMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50081499(4-Hydroxy-3-[(S)-2-oxo-3-(thieno[2,3-c]pyridine-2-...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against plasmin in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50289436((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration of the compound against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50289434((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50: <25nMAssay Description:Inhibitory concentration against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50144535((2S,3R)-4-Oxo-1-[4-(6-phenyl-hexanoyl)-piperazine-...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50144551((2S,3R)-1-(4-tert-Butylcarbamoyl-piperazine-1-carb...)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50076219((3S,6R)-6-Amino-6-benzyl-octahydro-indolizine-3-ca...)
Affinity DataIC50:  251nMAssay Description:Inhibitory concentration of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50144532((2S,3R)-4-Oxo-1-[4-(6-phenyl-hexanoyl)-piperazine-...)
Affinity DataIC50:  309nMAssay Description:Inhibitory activity of compound against Plasmin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
The Procter & Gamble

Curated by ChEMBL
LigandPNGBDBM50144555((R)-1-{4-[2-(4-Benzyloxy-phenyl)-acetyl]-piperazin...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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