Compile Data Set for Download or QSAR
Report error Found 8 of affinity data for UniProtKB/TrEMBL: P16519
TargetNeuroendocrine convertase 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446944BDBM50446944(CHEMBL3115771)
Affinity DataKi:  0.240nMAssay Description:Inhibition of human PC2 expressed in drosophila schneider 2 cells using pyroGlu-Arg-Thr-Lys-Arg-AMC as substrate after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuroendocrine convertase 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533413BDBM50533413(CHEMBL3126388)
Affinity DataKi:  0.360nMAssay Description:Inhibition of recombinant C-terminal truncated human SPC2 expressed in drosophila Schneider 2 cells after 1 hr by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNeuroendocrine convertase 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446945BDBM50446945(CHEMBL3115770)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human PC2 expressed in drosophila schneider 2 cells using pyroGlu-Arg-Thr-Lys-Arg-AMC as substrate after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuroendocrine convertase 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303776BDBM50303776(N-((6S,9S,12S)-1,17-diamino-6-(4-carbamimidoylbenz...)
Affinity DataKi:  55nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeuroendocrine convertase 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303774BDBM50303774(phenylacetyl-Arg-Val-Arg-4-amidinobenzylamide | CH...)
Affinity DataKi:  312nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeuroendocrine convertase 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303775BDBM50303775((S)-2-acetamido-N-((S)-1-((S)-1-(4-carbamimidoylbe...)
Affinity DataKi:  1.39E+3nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeuroendocrine convertase 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303777BDBM50303777((S)-5-guanidino-N-((S)-1-((S)-5-guanidino-1-(3-gua...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeuroendocrine convertase 2(Human)
University of Sherbrooke

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303778BDBM50303778((S)-N-((1-carbamimidoylpiperidin-4-yl)methyl)-5-gu...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed