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TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.0320nMAssay Description:Displacement of [125I]somatostatin from human SSTR3 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM85323(LTT-SRIF28 | SRIF28-Leu8,D-Trp22,Tyr25)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.140nMAssay Description:Inhibition of human sst3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM85323(LTT-SRIF28 | SRIF28-Leu8,D-Trp22,Tyr25)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50054462(CHEMBL3323076)
Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at human SSTR3 expressed in CHO cells assessed as cAMP level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476134(CHEMBL437296)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKd:  0.214nMAssay Description:Binding assay at human somatostatin receptor 3 (hsst3) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50352489(CHEMBL1824052)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human sst3 receptor expressed in CCL39 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM523757(US11136312, Compound MM-I-87)
Affinity DataEC50:  0.249nMAssay Description:Measurement of forskolin stimulated inhibition of cAMP was performed via time-resolved fluorescence resonance energy transfer (TR-FRET) LANCE assay (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50019568(CHEMBL411836 | SRIF-14 | Somatostatin receptor lig...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.251nMAssay Description:Binding affinity towards human Somatostatin receptor type 3 (sst3) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM523756(US11136312, Compound MM-I-83)
Affinity DataEC50:  0.276nMAssay Description:Measurement of forskolin stimulated inhibition of cAMP was performed via time-resolved fluorescence resonance energy transfer (TR-FRET) LANCE assay (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50091509(CHEMBL3582344)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity against human recombinant SSTR3 expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50474235(CHEMBL3349606)
Affinity DataKi:  0.316nMAssay Description:Binding affinity towards human Somatostatin receptor type 3 (sst3) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476138(CHEMBL376485)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50352480(CHEMBL1824051)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at human sst3 receptor expressed in CCL39 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM82467(CGP-23996 | 2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-...)
Affinity DataKi:  0.390nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50091513(CHEMBL3582321)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity against human recombinant SSTR3 expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50091503(CHEMBL3582339)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity against human recombinant SSTR3 expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50154508(CHEMBL3775042)
Affinity DataEC50:  0.460nMAssay Description:Antagonist activity at human somatostatin receptor type 3 assessed as inhibition of cAMP levelsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2017
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50212467(Sandostatinm)
Affinity DataIC50: 0.460nMAssay Description:Compound was tested for free energy of binding against somatostatin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2018
Entry Details

TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM84989(SS-25)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50091507(CHEMBL3582342)
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity against human recombinant SSTR3 expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476142(CHEMBL376484)
Affinity DataIC50: 0.5nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
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