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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
 
Diphenylborinic acid is a strong inhibitor of serine proteasesEBI
TBA
Potent Lys Patch-Containing Stapled Peptides Targeting PCSK9.EBI
Universit£
Bioactive Cyclization Optimizes the Affinity of a Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) Peptide Inhibitor.EBI
The University of Queensland
Discovery of Small-Molecule CD33 Pre-mRNA Splicing Modulators.EBI
Pfizer
A Series of Novel, Highly Potent, and Orally Bioavailable Next-Generation Tricyclic Peptide PCSK9 Inhibitors.EBI
Merck
From methylene bridged diindole to carbonyl linked benzimidazoleindole: Development of potent and metabolically stable PCSK9 modulators.EBI
University of Wisconsin-Madison
Series of Novel and Highly Potent Cyclic Peptide PCSK9 Inhibitors Derived from an mRNA Display Screen and Optimized via Structure-Based Design.EBI
Merck
Novel Cyclic Tetramer Compounds as PCSK9 Inhibitors for Treating Metabolic Disorders.EBI
Lauren Mccallister
Discovery of 2,3'-diindolylmethanes as a novel class of PCSK9 modulators.EBI
University of Wisconsin
Small molecules as inhibitors of PCSK9: Current status and future challenges.EBI
China Pharmaceutical University
Small molecule modulators of PCSK9 - A literature and patent overview.EBI
Astrazeneca
O'-(epoxyalkyl)tyrosines and (epoxyalkyl)phenylalanine as irreversible inactivators of serine proteases: synthesis and inhibition mechanism.EBI
State University