PMID

Data

Article Title

Organization

Identification and synthesis of [1,2,4]triazolo[3,4-a]phthalazine derivatives as high-affinity ligands to the alpha 2 delta-1 subunit of voltage gated calcium channel.

Merck Research Laboratories

Pyrazolopyridazine alpha-2-delta-1 ligands for the treatment of neuropathic pain.

Glaxosmithkline

Expedited SAR study of high-affinity ligands to the alpha(2)delta subunit of voltage-gated calcium channels: Generation of a focused library using a solution-phase Sn2Ar coupling methodology.

Merck Research Laboratories

N-Acridin-9-yl-butane-1,4-diamine derivatives: high-affinity ligands of the alpha2delta subunit of voltage gated calcium channels.

Merck Research Laboratories

Synthesis and biological evaluation of 6-aryl-6H-pyrrolo[3,4-d]pyridazine derivatives: high-affinity ligands to the alpha 2 delta subunit of voltage gated calcium channels.

Merck Research Laboratories

Piperazinyl Bicyclic Derivatives as Selective Ligands of the ?2?-1 Subunit of Voltage-Gated Calcium Channels.

Welab Barcelona

Bicyclic Diazepinones as Dual Ligands of the ?2?-1 Subunit of Voltage-Gated Calcium Channels and the Norepinephrine Transporter.

Esteve Pharmaceuticals

Structure-activity relationships of diphenylpiperazine N-type calcium channel inhibitors.

Neuromed Pharmaceuticals

Discovery of N-(5-Fluoropyridin-2-yl)-6-methyl-4-(pyrimidin-5-yloxy)picolinamide (VU0424238): A Novel Negative Allosteric Modulator of Metabotropic Glutamate Receptor Subtype 5 Selected for Clinical Evaluation.

Vanderbilt University Institute of Imaging Science