BindingDB

The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.5M data for 737K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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19 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification of novel GLUT inhibitors.EBI
Bayer Pharma
Oxime-based inhibitors of glucose transporter 1 displaying antiproliferative effects in cancer cells.EBI
University of Pisa
Development of a novel class of glucose transporter inhibitors.EBI
The Ohio State University
Discovery of canagliflozin, a novel C-glucoside with thiophene ring, as sodium-dependent glucose cotransporter 2 inhibitor for the treatment of type 2 diabetes mellitus.EBI
Mitsubishi Tanabe Pharma
Glucose promoiety enables glucose transporter mediated brain uptake of ketoprofen and indomethacin prodrugs in rats.EBI
University of Kuopio
Ovarian Cancer Relies on Glucose Transporter 1 to Fuel Glycolysis and Growth: Anti-Tumor Activity of BAY-876.EBI
Virginia Commonwealth University School of Medicine
GLUT4 expression and glucose transport in human induced pluripotent stem cell-derived cardiomyocytes.EBI
University of Glasgow
Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876.EBI
Bayer AG
NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family.EBI
Johann Wolfgang Goethe University
Interaction of O-(undec-10-en)-yl-D-glucose derivatives with the Plasmodium falciparum hexose transporter (PfHT).EBI
Université
Target Separation and Potential Anticancer Activity of Withanolide-Based Glucose Transporter Protein 1 Inhibitors from EBI
China Pharmaceutical University
Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential.EBI
Bharati Vidyapeeth'S College of Pharmacy
Discovery and Optimization of Glucose Uptake Inhibitors.EBI
Kadmon
The Druggability of Solute Carriers.EBI
The Scripps Research Institute
Monosaccharide Analogues of Anticancer Peptide R-Lycosin-I: Role of Monosaccharide Conjugation in Complexation and the Potential of Lung Cancer Targeting and Therapy.EBI
TBA
Development of GLUT4-selective antagonists for multiple myeloma therapy.EBI
Emory University
(Aminoalkyl)carbamates of forskolin: intermediates for the synthesis of functionalized derivatives of forskolin with different specificities for adenylyl cyclase and the glucose transporter.EBI
Food and Drug Administration
3′ end caps, 5′ end caps and combinations thereof for therapeutic RNABDB
Novartis
In vitro opioid activity profiles of 6-amino acid substituted derivatives of 14-O-methyloxymorphone.BDB
University of Innsbruck