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61 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Chemical and bioactivity of flavanones obtained from roots of Dalea pazensis Rusby.EBI
Universidad Nacional De C£Rdoba
2-Hydroxypyridine-EBI
Univ. Grenoble-Alpes/Cnrs
Bioactive Constituents of Glycyrrhiza uralensis (Licorice): Discovery of the Effective Components of a Traditional Herbal Medicine.EBI
Peking University
Rhododendrol glycosides as stereospecific tyrosinase inhibitors.EBI
Tokyo University of Agriculture and Technology
Effect of the tyrosinase inhibitor (S)-N-trans-feruloyloctopamine from garlic skin on tyrosinase gene expression and melanine accumulation in melanoma cells.EBI
Gansu College of Traditional Chinese Medicine
Structure-activity relationships of the thujaplicins for inhibition of human tyrosinase.EBI
Institute For Theoretical Medicine
Tyrosinase inhibitory activity of a glucosylated hydroxystilbene in mouse melan-a melanocytes.EBI
The Chinese University of Hong Kong
(-)-N-Formylanonaine from Michelia alba as a human tyrosinase inhibitor and antioxidant.EBI
Kaohsiung Medical University
New tyrosinase inhibitors selected by atomic linear indices-based classification models.EBI
Central University of Las Villas
Identification of oxidation product of arbutin in mushroom tyrosinase assay system.EBI
University of California
 
Synthesis of N-kojic-amino acid and N-kojic-amino acid-kojiate and their tyrosinase inhibitory activityEBI
TBA
New halogenated phenylcoumarins as tyrosinase inhibitors.EBI
Universidad De Santiago De Compostela
Synthesis and anti-melanogenic activity of hydroxyphenyl benzyl ether analogues.EBI
Catholic University of Daegu
Synthesis and evaluation of bibenzyl glycosides as potent tyrosinase inhibitors.EBI
Utsunomiya University
Natural ortho-dihydroxyisoflavone derivatives from aged Korean fermented soybean paste as potent tyrosinase and melanin formation inhibitors.EBI
Amorepacific
Evaluation of 3,4-dihydroquinazoline-2(1H)-thiones as inhibitors of alpha-MSH-induced melanin production in melanoma B16 cells.EBI
Chungnam National University
Synthesis and biological evaluation of curcumin-like diarylpentanoid analogues for anti-inflammatory, antioxidant and anti-tyrosinase activities.EBI
Universiti Putra Malaysia
N-[(Dihydroxyphenyl)acyl]serotonins as potent inhibitors of tyrosinase from mouse and human melanoma cells.EBI
National Institute of Advanced Industrial Science and Technology
Biphenyl glycosides from the fruit of Pyracantha fortuneana.EBI
Shenyang Pharmaceutical University
Constituents from the leaves of Phellodendron amurense var. wilsonii and their bioactivity.EBI
National Cheng Kung University
Acetophenone derivatives from Acronychia pedunculata.EBI
National Cheng Kung University
Catechol-mimicking transition-state analogues as non-oxidizable inhibitors of tyrosinases.EBI
Univ. Grenoble Alpes
Computational methods to analyze and predict the binding mode of inhibitors targeting both human and mushroom tyrosinase.EBI
University of Messina
The recent discovery of a promising pharmacological scaffold derived from carvacrol: A review.EBI
Universiti Kebangsaan Malaysia
Synthesis and evaluation of 3-hydroxyquinolin-2(1H)-one derivatives as inhibitors of tyrosinase.EBI
North-West University
Pyrrole-containing hybrids as potential anticancer agents: An insight into current developments and structure-activity relationships.EBI
Jiangxi Science & Technology Normal University
Recent advances in triazoles as tyrosinase inhibitors.EBI
University of Health Sciences
Artificial Intelligence-Assisted Optimization of Antipigmentation Tyrosinase Inhibitors: De Novo Molecular Generation Based on a Low Activity Lead Compound.EBI
Hangzhou Normal University
Design and synthesis of 4-amino-2',4'-dihydroxyindanone derivatives as potent inhibitors of tyrosinase and melanin biosynthesis in human melanoma cells.EBI
University of Grenoble Alpes
Synthetic tyrosyl gallate derivatives as potent melanin formation inhibitors.EBI
Amorepacific
Resorcinol-based hemiindigoid derivatives as human tyrosinase inhibitors and melanogenesis suppressors in human melanoma cells.EBI
University Grenoble Alpes
Azole inhibitors of mushroom and human tyrosinases: Current advances and prospects of drug development for melanogenic dermatological disorders.EBI
King Saud University
Exploiting HOPNO-dicopper center interaction to development of inhibitors for human tyrosinase.EBI
University of Grenoble Alpes
Recent advances in the design and discovery of synthetic tyrosinase inhibitors.EBI
National Clinical Research Center For Geriatrics
Pyrazolotriazines: Biological activities, synthetic strategies and recent developments.EBI
Mazandaran University of Medical Sciences
Tyrosinase inhibitors as potential antibacterial agents.EBI
The University of Queensland
Chemical transformations of oxyresveratrol (trans-2,4,3',5'-tetrahydroxystilbene) into a potent tyrosinase inhibitor and a strong cytotoxic agent.EBI
Chulalongkorn University
Discovery of benzylidenebenzofuran-3(2H)-one (aurones) as inhibitors of tyrosinase derived from human melanocytes.EBI
Umr-Cnrs 5063
Polyphenolic compounds: Synthesis, assessment of antimicrobial effect and enzymes inhibition against important medicinal enzymes with computational details.EBI
Bartin University
Design, synthesis and biological evaluation of tyrosinase-targeting PROTACs.EBI
University of Chinese Academy of Sciences
Solid-phase synthesis of kojic acid-tripeptides and their tyrosinase inhibitory activity, storage stability, and toxicity.EBI
Seoul National University
2-hydroxy-4-isopropylbenzaldehyde, a potent partial tyrosinase inhibitor.EBI
University of California
Kojic acid-natural product conjugates as mushroom tyrosinase inhibitors.EBI
Mazandaran University of Medical Sciences
Advances in the Design of Genuine Human Tyrosinase Inhibitors for Targeting Melanogenesis and Related Pigmentations.EBI
Universite Grenoble Alpes
Xanthones for melanogenesis inhibition: Molecular docking and QSAR studies to understand their anti-tyrosinase activity.EBI
Universidade Dos A£Ores
Aurone: A biologically attractive scaffold as anticancer agent.EBI
King Khalid University
Recent applications of hydantoin and thiohydantoin in medicinal chemistry.EBI
College of Pharmacy and Gachon Institute of Pharmaceutical Science
Inhibitors of Melanogenesis: An Updated Review.EBI
University of Bonn
Insights into the chemistry and therapeutic potential of furanones: A versatile pharmacophore.EBI
Jamia Hamdard
Isolation of Sesquiterpene-Amino Acid Conjugates, Onopornoids A-D, and a Flavonoid Glucoside from Onopordum alexandrinum.EBI
Hiroshima University
Melanogenic inhibitory effects of Triangularin in B16F0 melanoma cells, in vitro and molecular docking studies.EBI
Universidad Nacional De C£Rdoba
Dimeric cinnamoylamide analogues for regulation of tyrosinase activity in melanoma cells: A role of diamide-link chain length.EBI
Seoul National University of Science and Technology
Resorcinol alkyl glucosides as potent tyrosinase inhibitors.EBI
Utsunomiya University
Refinement of the pharmacophore of 3,4-dihydroquinazoline-2(1H)-thiones for their anti-melanogenesis activity.EBI
Chungnam National University
Targeting Tyrosinase: Development and Structural Insights of Novel Inhibitors Bearing Arylpiperidine and Arylpiperazine Fragments.EBI
Universit�
Artocarmins G-M, Prenylated 4-Chromenones from the Stems of Artocarpus rigida and Their Tyrosinase Inhibitory Activities.EBI
Hiroshima University
Glycybridins A-K, Bioactive Phenolic Compounds from Glycyrrhiza glabra.EBI
Peking University
Pyridone derivative, pharmaceutical containing the same and methods of use thereofBDB
Kaken Pharmaceutical
Benzolamide is not a membrane-impermeant carbonic anhydrase inhibitor.BDB
UniversitÀ Degli Studi Di Firenze