186 articles for thisTarget
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Chemical and bioactivity of flavanones obtained from roots of Dalea pazensis Rusby.
Universidad Nacional De C£Rdoba
Synthesis and biological evaluation of novel hydroxybenzaldehyde-based kojic acid analogues as inhibitors of mushroom tyrosinase.
Hunan University of Science and Technology
Design and synthesis of novel hydroxypyridinone derivatives as potential tyrosinase inhibitors.
Zhejiang Gongshang University
Bioactive Constituents of Glycyrrhiza uralensis (Licorice): Discovery of the Effective Components of a Traditional Herbal Medicine.
Peking University
N-Acyl Dehydrotyrosines, Tyrosinase Inhibitors from the Marine Bacterium Thalassotalea sp. PP2-459.
University of Rhode Island
Design and synthesis of thiourea derivatives with sulfur-containing heterocyclic scaffolds as potential tyrosinase inhibitors.
East China University of Science and Technology
Identification of six new lupane-type triterpenoids from Acanthopanax koreanum leaves and their tyrosinase inhibitory activities.
Catholic University of Daegu
One-pot green synthesis of 1,3,5-triarylpentane-1,5-dione and triarylmethane derivatives as a new class of tyrosinase inhibitors.
Jiangnan University
Highly potent tyrosinase inhibitor, neorauflavane from Campylotropis hirtella and inhibitory mechanism with molecular docking.
Gyeongsang National University
Inhibitory kinetics of novel 2,3-dihydro-1H-inden-1-one chalcone-like derivatives on mushroom tyrosinase.
University of Technology Sydney
Design and synthesis of aloe-emodin derivatives as potent anti-tyrosinase, antibacterial and anti-inflammatory agents.
Shaoyang University
Synthesis of novel compounds containing morpholine and 5(4H)-oxazolone rings as potent tyrosinase inhibitors.
Payame Noor University (Pnu)
Integrated kinetic studies and computational analysis on naphthyl chalcones as mushroom tyrosinase inhibitors.
University of Technology Sydney
Rhododendrol glycosides as stereospecific tyrosinase inhibitors.
Tokyo University of Agriculture and Technology
Synthesis, kinetic mechanism and docking studies of vanillin derivatives as inhibitors of mushroom tyrosinase.
Kongju National University
Inhibitors of melanogenesis in B16 melanoma 4A5 cells from flower buds of Lawsonia inermis (Henna).
Kyoto Pharmaceutical University
Structure-based modification of 3-/4-aminoacetophenones giving a profound change of activity on tyrosinase: from potent activators to highly efficient inhibitors.
Sun Yat-Sen University
Azachalcones: a new class of potent polyphenol oxidase inhibitors.
University of Technology Sydney
Effect of the tyrosinase inhibitor (S)-N-trans-feruloyloctopamine from garlic skin on tyrosinase gene expression and melanine accumulation in melanoma cells.
Gansu College of Traditional Chinese Medicine
Rational design, synthesis and structure-activity relationships of 4-alkoxy- and 4-acyloxy-phenylethylenethiosemicarbazone analogues as novel tyrosinase inhibitors.
Sun Yat-Sen University
Bioactive benzofuran derivatives: moracins A-Z in medicinal chemistry.
Dongguk University-Seoul
Flavokawains B and C, melanogenesis inhibitors, isolated from the root of Piper methysticum and synthesis of analogs.
Sungkyunkwan University
Structure-activity relationships of the thujaplicins for inhibition of human tyrosinase.
Institute For Theoretical Medicine
Anti-tyrosinase, antioxidant, and antibacterial activities of novel 5-hydroxy-4-acetyl-2,3-dihydronaphtho[1,2-b]furans.
Yeungnam University
Tyrosinase inhibitory activity of a glucosylated hydroxystilbene in mouse melan-a melanocytes.
The Chinese University of Hong Kong
Synthesis, biological evaluation, and molecular docking of N-{3-[3-(9-methyl-9H-carbazol-3-yl)-acryloyl]-phenyl}-benzamide/amide derivatives as xanthine oxidase and tyrosinase inhibitors.
Solapur University
Synthesis and biological evaluation of a novel series of bis-salicylaldehydes as mushroom tyrosinase inhibitors.
Universit£
(-)-N-Formylanonaine from Michelia alba as a human tyrosinase inhibitor and antioxidant.
Kaohsiung Medical University
Synthesis and biological evaluation of novel 4-hydroxybenzaldehyde derivatives as tyrosinase inhibitors.
Sun Yat-Sen University
Synthesis and evaluation of 5-benzylidene(thio)barbiturate-beta-D-glycosides as mushroom tyrosinase inhibitors.
Sun Yat-Sen University
Analogues of N-hydroxy-N'-phenylthiourea and N-hydroxy-N'-phenylurea as inhibitors of tyrosinase and melanin formation.
Mayoly Spindler
1-(1-Arylethylidene)thiosemicarbazide derivatives: a new class of tyrosinase inhibitors.
Sun Yat-Sen University
Dragon method for finding novel tyrosinase inhibitors: Biosilico identification and experimental in vitro assays.
Central University of Las Villas
New tyrosinase inhibitors selected by atomic linear indices-based classification models.
Central University of Las Villas
Identification of oxidation product of arbutin in mushroom tyrosinase assay system.
University of California
Synthesis of N-kojic-amino acid and N-kojic-amino acid-kojiate and their tyrosinase inhibitory activity
TBA
2-Arylbenzofuran, flavonoid, and tyrosinase inhibitory constituents of Morus yunnanensis.
Fudan University
Molecular docking studies of a phlorotannin, dieckol isolated from Ecklonia cava with tyrosinase inhibitory activity.
Jeju National University
Inhibitory activity of novel kojic acid derivative containing trolox moiety on melanogenesis.
Kyung Hee University Skin Biotechnology Center
Structural requirement of phenylthiourea analogs for their inhibitory activity of melanogenesis and tyrosinase.
Chungnam National University
Refinement of arylthiosemicarbazone pharmacophore in inhibition of mushroom tyrosinase.
Universit£
Gusanlungionosides A-D, potential tyrosinase inhibitors from Arcangelisia gusanlung.
Institute of Medicinal Plant Development
New halogenated phenylcoumarins as tyrosinase inhibitors.
Universidad De Santiago De Compostela
Synthesis and anti-melanogenic activity of hydroxyphenyl benzyl ether analogues.
Catholic University of Daegu
Synthesis and structure-activity relationships of phenylpropanoid amides of serotonin on tyrosinase inhibition.
Kinki University
Synthesis and evaluation of bibenzyl glycosides as potent tyrosinase inhibitors.
Utsunomiya University
Evaluation of dihydropyrimidin-(2H)-one analogues and rhodanine derivatives as tyrosinase inhibitors.
Shaoyang University
Synthesis and biological activity of hydroxy substituted phenyl-benzo[d]thiazole analogues for antityrosinase activity in B16 cells.
Pusan National University
Prenylated flavanones with anti-tyrosinase activity from Dalea boliviana.
Universidad Nacional De Co£?Rdoba
Benzyl benzoates: New phlorizin analogs as mushroom tyrosinase inhibitors.
Sun Yat-Sen University
Identifying chelators for metalloprotein inhibitors using a fragment-based approach.
University of California
Changes in flavonoid content and tyrosinase inhibitory activity in kenaf leaf extract after far-infrared treatment.
Amorepacific
A novel ring-expanded product with enhanced tyrosinase inhibitory activity from classical Fe-catalyzed oxidation of rosmarinic acid, a potent antioxidative Lamiaceae polyphenol.
University of Tokushima
Structural insights into the hot spot amino acid residues of mushroom tyrosinase for the bindings of thujaplicins.
Institute For Theoretical Medicine
Kojyl thioether derivatives having both tyrosinase inhibitory and anti-inflammatory properties.
Amorepacific
Design and synthesis of biphenyl derivatives as mushroom tyrosinase inhibitors.
Jinan University
Synthesis of novel 3,5-diaryl pyrazole derivatives using combinatorial chemistry as inhibitors of tyrosinase as well as potent anticancer, anti-inflammatory agents.
Solapur University
A newly synthesized, potent tyrosinase inhibitor: 5-(6-hydroxy-2-naphthyl)-1,2,3-benzenetriol.
Pusan National University
Alpneumines A-H, new anti-melanogenic indole alkaloids from Alstonia pneumatophora.
Hoshi University
New potent inhibitors of tyrosinase: novel clues to binding of 1,3,4-thiadiazole-2(3H)-thiones, 1,3,4-oxadiazole-2(3H)-thiones, 4-amino-1,2,4-triazole-5(4H)-thiones, and substituted hydrazides to the dicopper active site.
King Saud University
Synthesis and biological activity of oxadiazole and triazolothiadiazole derivatives as tyrosinase inhibitors.
University Putra Malaysia
Evaluation of anti-pigmentary effect of synthetic sulfonylamino chalcone.
Department of Functional Crop
Tyrosinase-inhibitory constituents from the twigs of Cinnamomum cassia.
Chungnam National University
Asymmetric syntheses of daedalin A and quercinol and their tyrosinase inhibitory activity.
Shinshu University
Natural ortho-dihydroxyisoflavone derivatives from aged Korean fermented soybean paste as potent tyrosinase and melanin formation inhibitors.
Amorepacific
Melanogenesis inhibitors from the desert plant Anastatica hierochuntica in B16 melanoma cells.
Kyoto Pharmaceutical University
Evaluation of 3,4-dihydroquinazoline-2(1H)-thiones as inhibitors of alpha-MSH-induced melanin production in melanoma B16 cells.
Chungnam National University
Melanogenesis inhibitors from the rhizomes of Alpinia officinarum in B16 melanoma cells.
Kyoto Pharmaceutical University
Discovery of 4-functionalized phenyl-O-beta-D-glycosides as a new class of mushroom tyrosinase inhibitors.
Sun Yat-Sen University
Inhibitory effects of 5-benzylidene barbiturate derivatives on mushroom tyrosinase and their antibacterial activities.
Sun Yat-Sen University
Antityrosinase and Antioxidant Effects of ent-Kaurane Diterpenes from Leaves of Broussonetia papyrifera.
Tajen University
Synthesis and biological evaluation of curcumin-like diarylpentanoid analogues for anti-inflammatory, antioxidant and anti-tyrosinase activities.
Universiti Putra Malaysia
N-[(Dihydroxyphenyl)acyl]serotonins as potent inhibitors of tyrosinase from mouse and human melanoma cells.
National Institute of Advanced Industrial Science and Technology
Potential antioxidants and tyrosinase inhibitors from synthetic polyphenolic deoxybenzoins.
National Taiwan University
Studies on depigmenting activities of dihydroxyl benzamide derivatives containing adamantane moiety.
Amorepacific
PEG-immobilization of cardol and soluble polymer-supported synthesis of some cardol-coumarin derivatives: preliminary evaluation of their inhibitory activity on mushroom tyrosinase.
Università
Tyrosinase inhibitory effects of 1,3-diphenylpropanes from Broussonetia kazinoki.
Graduate School of Gyeongsang National University
Synthesis of tyrosinase inhibitory (4-oxo-4H-pyran-2-yl)acrylic acid ester derivatives.
Institute of Science and Technology
Synthesis and biological evaluation of helicid analogues as mushroom tyrosinase inhibitors.
Sun Yat-Sen University
Molecular design of potent tyrosinase inhibitors having the bibenzyl skeleton.
Utsunomiya University
A class of potent tyrosinase inhibitors: alkylidenethiosemicarbazide compounds.
Sun Yat-Sen University
Pyronane monoterpenoids from the fruit of Gardenia jasminoides.
Chungnam National University
Complex sesquiterpenoids with tyrosinase inhibitory activity from the leaves of Chloranthus tianmushanensis.
Zhejiang University
Biphenyl glycosides from the fruit of Pyracantha fortuneana.
Shenyang Pharmaceutical University
Antityrosinase principles and constituents of the petals of Crocus sativus.
National Cheng Kung University
Constituents from the leaves of Phellodendron amurense var. wilsonii and their bioactivity.
National Cheng Kung University
Constituents of the stigmas of Crocus sativus and their tyrosinase inhibitory activity.
National Cheng Kung University
A new dimeric stilbene with tyrosinase inhibitiory activity from Artocarpus gomezianus.
Chulalongkorn University
Discovery of small-molecule inhibitors of tyrosinase.
University of Texas Southwestern Medical Center
Synthetic tyrosyl gallate derivatives as potent melanin formation inhibitors.
Amorepacific
Enhanced substituted resorcinol hydrophobicity augments tyrosinase inhibition potency.
Migal - Galilee Technology Center
Synthesis and evaluation of 2',4',6'-trihydroxychalcones as a new class of tyrosinase inhibitors.
Hokkaido University
Modulating effects of a novel skin-lightening agent, alpha-lipoic acid derivative, on melanin production by the formation of DOPA conjugate products.
Dhc
Inhibitory effects of phloridzin dihydrate on the activity of mushroom (Agaricus bisporus) tyrosinase.
Xiamen University
TOMOCOMD-CARDD descriptors-based virtual screening of tyrosinase inhibitors: evaluation of different classification model combinations using bond-based linear indices.
Central University of Las Villas
Recent advances in the design and discovery of synthetic tyrosinase inhibitors.
National Clinical Research Center For Geriatrics
Pyrazolotriazines: Biological activities, synthetic strategies and recent developments.
Mazandaran University of Medical Sciences
Syntheses of hydroxy substituted 2-phenyl-naphthalenes as inhibitors of tyrosinase.
Pusan National University
Bioactive Aurones, Indanones, and Other Hemiindigoid Scaffolds: Medicinal Chemistry and Photopharmacology Perspectives.
Universite Grenoble Alpes
An overview of hydroxypyranone and hydroxypyridinone as privileged scaffolds for novel drug discovery.
Guizhou Medical University
A medicinal chemistry perspective of drug repositioning: Recent advances and challenges in drug discovery.
University of Bonn
Chemical transformations of oxyresveratrol (trans-2,4,3',5'-tetrahydroxystilbene) into a potent tyrosinase inhibitor and a strong cytotoxic agent.
Chulalongkorn University
N-Benzylbenzamides: a new class of potent tyrosinase inhibitors.
Seoul National University
Discovery of benzylidenebenzofuran-3(2H)-one (aurones) as inhibitors of tyrosinase derived from human melanocytes.
Umr-Cnrs 5063
Polyphenolic compounds: Synthesis, assessment of antimicrobial effect and enzymes inhibition against important medicinal enzymes with computational details.
Bartin University
Design, synthesis and biological evaluation of tyrosinase-targeting PROTACs.
University of Chinese Academy of Sciences
Solid-phase synthesis of kojic acid-tripeptides and their tyrosinase inhibitory activity, storage stability, and toxicity.
Seoul National University
2-hydroxy-4-isopropylbenzaldehyde, a potent partial tyrosinase inhibitor.
University of California
Kojic acid-natural product conjugates as mushroom tyrosinase inhibitors.
Mazandaran University of Medical Sciences
Novel 1,3,4-oxadiazole compounds inhibit the tyrosinase and melanin level: Synthesis, in-vitro, and in-silico studies.
Kongju National University
Advances in the Design of Genuine Human Tyrosinase Inhibitors for Targeting Melanogenesis and Related Pigmentations.
Universit£
Xanthones for melanogenesis inhibition: Molecular docking and QSAR studies to understand their anti-tyrosinase activity.
Universidade Dos A£Ores
Recent applications of hydantoin and thiohydantoin in medicinal chemistry.
College of Pharmacy and Gachon Institute of Pharmaceutical Science
2-(4-Fluorophenyl)-quinazolin-4(3H)-one as a novel tyrosinase inhibitor: Synthesis, inhibitory activity, and mechanism.
Jiangxi Normal University
Synthesis and bioactivity of novel isoxazole chalcone derivatives on tyrosinase and melanin synthesis in murine B16 cells for the treatment of vitiligo.
Chinese Academy of Sciences
Discovery of a new type of scaffold for the creation of novel tyrosinase inhibitors.
Hinoki Shinyaku
Benzo[b]thiophene-thiazoles as potent anti-Toxoplasma gondii agents: Design, synthesis, tyrosinase/tyrosine hydroxylase inhibitors, molecular docking study, and antioxidant activity.
Nicolaus Copernicus University
Insights on the synthesis of asymmetric curcumin derivatives and their biological activities.
Universiti Kuala Lumpur
Tyrosinase inhibitory study of flavonolignans from the seeds of Silybum marianum (Milk thistle).
Gyeongsang National University
Synthesis of N-hydroxycinnamoyl amide derivatives and evaluation of their anti-oxidative and anti-tyrosinase activities.
Beijing Technology and Business University
Insights into the chemistry and therapeutic potential of furanones: A versatile pharmacophore.
Jamia Hamdard
Isolation of Sesquiterpene-Amino Acid Conjugates, Onopornoids A-D, and a Flavonoid Glucoside from Onopordum alexandrinum.
Hiroshima University
Veratric acid derivatives containing benzylidene-hydrazine moieties as promising tyrosinase inhibitors and free radical scavengers.
Shiraz University of Medical Sciences
Melanogenic inhibitory effects of Triangularin in B16F0 melanoma cells, in vitro and molecular docking studies.
Universidad Nacional De C£Rdoba
Dimeric cinnamoylamide analogues for regulation of tyrosinase activity in melanoma cells: A role of diamide-link chain length.
Seoul National University of Science and Technology
Exploiting the 1-(4-fluorobenzyl)piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and biological profile.
Polo Universitario Ss. Annunziata
Discovery of tropinone-thiazole derivatives as potent caspase 3/7 activators, and noncompetitive tyrosinase inhibitors with high antiproliferative activity: Rational design, one-pot tricomponent synthesis, and lipophilicity determination.
Nicolaus Copernicus University
Hydroxyl substituted benzoic acid/cinnamic acid derivatives: Tyrosinase inhibitory kinetics, anti-melanogenic activity and molecular docking studies.
The University of Queensland (Uq)
Synthesis of cinnamic amide derivatives and their anti-melanogenic effect in ?-MSH-stimulated B16F10 melanoma cells.
Pusan National University
De Novo Molecular Design of a Novel Octapeptide That Inhibits In Vivo Melanogenesis and Has Great Transdermal Ability.
Dalian University of Technology
From bench to counter: Discovery and validation of a peony extract as tyrosinase inhibiting cosmeceutical.
University of Innsbruck
Synthesis and tyrosinase inhibitory activities of 4-oxobutanoate derivatives of carvacrol and thymol.
Susquehanna University
Analogues of ethionamide, a drug used for multidrug-resistant tuberculosis, exhibit potent inhibition of tyrosinase.
Kyungpook National University
Design, synthesis and biological evaluation of hydroxy- or methoxy-substituted 5-benzylidene(thio) barbiturates as novel tyrosinase inhibitors.
China National Analytical Center (Guangzhou)
Inhibitory effects of novel synthetic methimazole derivatives on mushroom tyrosinase and melanogenesis.
Hungkuang University
Inhibition of tyrosinase activity by polyphenol compounds from Flemingia philippinensis roots.
Gyeongsang National University
Chemical synthesis and tyrosinase inhibitory activity of rhododendrol glycosides.
Tokyo University of Agriculture and Technology
Synthesis, antioxidant capacity, and structure-activity relationships of tri-O-methylnorbergenin analogues on tyrosinase inhibition.
Kinki University
De novo tyrosinase inhibitor: 4-(6,7-dihydro-5H-indeno[5,6-d]thiazol-2-yl)benzene-1,3-diol (MHY1556).
Pusan National University
Synthesis of new heterocyclic hybrids based on pyrazole and thiazolidinone scaffolds as potent inhibitors of tyrosinase.
Bahirji Smarak Mahavidyalaya
Synthesis of novel azo compounds containing 5(4H)-oxazolone ring as potent tyrosinase inhibitors.
Payame Noor University
Design and synthesis of 3,5-diaryl-4,5-dihydro-1H-pyrazoles as new tyrosinase inhibitors.
Sun Yat-Sen University
Synthesis and dual biological effects of hydroxycinnamoyl phenylalanyl/prolyl hydroxamic acid derivatives as tyrosinase inhibitor and antioxidant.
Seoul National University
Synthesis and antityrosinase activities of alkyl 3,4-dihydroxybenzoates.
Xiamen University
Neonicotinoid insecticides: oxidative stress in planta and metallo-oxidase inhibition.
University of California
Synthesis of novel azo-resveratrol, azo-oxyresveratrol and their derivatives as potent tyrosinase inhibitors.
Pusan National University
Design, synthesis and molecular simulation studies of dihydrostilbene derivatives as potent tyrosinase inhibitors.
University of Athens
Tyrosinase inhibitory activity of a 6-isoprenoid-substituted flavanone isolated from Dalea elegans.
Catholic University of C£Rdoba
Design and synthesis of 5-(substituted benzylidene)thiazolidine-2,4-dione derivatives as novel tyrosinase inhibitors.
Pusan National University
Depigmenting activities of kojic acid derivatives without tyrosinase inhibitory activities.
Hanyang University
Depigmenting activity of new kojic acid derivative obtained as a side product in the synthesis of cinnamate of kojic acid.
Hanyang University
Adamantyl N-benzylbenzamide: new series of depigmentation agents with tyrosinase inhibitory activity.
Amorepacific Corporation R&D Center
Refinement of the pharmacophore of 3,4-dihydroquinazoline-2(1H)-thiones for their anti-melanogenesis activity.
Chungnam National University
The tyrosinase inhibitory effects of isoxazolone derivatives with a (Z)-?-phenyl-?, ?-unsaturated carbonyl scaffold.
Pusan National University
Targeting Tyrosinase: Development and Structural Insights of Novel Inhibitors Bearing Arylpiperidine and Arylpiperazine Fragments.
Universit�
Design, synthesis, kinetic mechanism and molecular docking studies of novel 1-pentanoyl-3-arylthioureas as inhibitors of mushroom tyrosinase and free radical scavengers.
Quaid-I-Azam University
Artocarmins G-M, Prenylated 4-Chromenones from the Stems of Artocarpus rigida and Their Tyrosinase Inhibitory Activities.
Hiroshima University
Isolation of Flavonoids and Flavonoid Glycosides from Myrsine africana and Their Inhibitory Activities against Mushroom Tyrosinase.
University of Pretoria
Study on the design, synthesis and structure-activity relationships of new thiosemicarbazone compounds as tyrosinase inhibitors.
Sun Yat-Sen University
Developing hybrid molecule therapeutics for diverse enzyme inhibitory action: Active role of coumarin-based structural leads in drug discovery.
Abbottabad University of Science and Technology
Glycybridins A-K, Bioactive Phenolic Compounds from Glycyrrhiza glabra.
Peking University
Molecular docking studies and biological evaluation of 1,3,4-thiadiazole derivatives bearing Schiff base moieties as tyrosinase inhibitors.
Shaoyang University
Synthesis and tyrosinase inhibition activity of trans-stilbene derivatives.
Indian Institute of Integrative Medicine
Synthesis and biological evaluation of kojic acid derivatives containing 1,2,4-triazole as potent tyrosinase inhibitors.
Hunan University of Science and Technology
Microwave-assisted synthesis and tyrosinase inhibitory activity of chalcone derivatives.
Shaoyang University
Inhibitory effects on mushroom tyrosinase by flavones from the stem barks of Morus lhou (S.) Koidz.
Gyeongsang National University
Effects of hydroxybenzyl alcohols on melanogenesis in melanocyte-keratinocyte co-culture and monolayer culture of melanocytes.
National Tsing Hua University
The inhibitory effect of some new synthesized xanthates on mushroom tyrosinase activities.
University of Tehran
Tyrosinase inhibition: conformational analysis based studies on molecular dynamics calculations of bipiperidine based inhibitors.
University of Karachi