Target Names are taken from UniProtKB. To view the associated UniProt page, click on the UniProt ID. When we have data for a given Target in multiple species or for mutants of a given Target, we provide a header row (upper case, bold font) with all of the data followed by a separate for each species or variant of the Target.
Target Name
Organism
Affinity Links
Articles
UniProts
Files
Human
Escherichia coli K-12 (Enterobacteria)
Mycobacterium tuberculosis
Escherichia coli O127:H6 (strain E2348/69 / EPEC)
Ki: 3
Haemophilus influenzae (strain 86-028NP)
Human
Mus musculus (mouse)
Rattus norvegicus (rat)
Mus musculus (mouse)
Rattus norvegicus
Escherichia coli (strain K12)
IC50: 4
Escherichia coli (Enterobacteria)
Ki: 1
Human
Rattus norvegicus
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/catalytic subunit alpha-2/subunit beta-1/subunit beta-2/subunit gamma-1/subunit gamma-2/subunit gamma-3 O54950 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078
Mus musculus
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1 P54619 Q13131 Q9Y478
Human
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-2 Q13131 Q9UGJ0 Q9Y478
Human
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-3 Q13131 Q9UGI9 Q9Y478
Human
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-2/subunit gamma-1 P54645 P80385 Q9QZH4
Rattus norvegicus
EC50: 3
5'-AMP-activated protein kinase catalytic subunit alpha-1/catalytic subunit alpha-2/subunit beta-1/subunit beta-2/subunit gamma-1/subunit gamma-2/subunit gamma-3 O54950 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078
Mus musculus
EC50: 1
Human
Rattus norvegicus
EC50: 3
5'-AMP-activated protein kinase catalytic subunit alpha-2/subunit beta-1/subunit gamma-1 P54619 P54646 Q9Y478
Human
5'-AMP-activated protein kinase catalytic subunit alpha-1/catalytic subunit alpha-2/subunit beta-1/subunit beta-2/subunit gamma-1/subunit gamma-2/subunit gamma-3 O54950 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078
Mus musculus
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1 P54619 Q13131 Q9Y478
Human
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-2 Q13131 Q9UGJ0 Q9Y478
Human
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-3 Q13131 Q9UGI9 Q9Y478
Human
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-2/subunit beta-1/subunit gamma-1 P54619 P54646 Q9Y478
Human
5'-AMP-activated protein kinase catalytic subunit alpha-1/catalytic subunit alpha-2/subunit beta-1/subunit beta-2/subunit gamma-1/subunit gamma-2/subunit gamma-3 O54950 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078
Mus musculus
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-2/subunit gamma-1 P54645 P80385 Q9QZH4
Rattus norvegicus
EC50: 3
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-2/subunit gamma-1 O43741 P54619 Q13131
Human
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-2/subunit gamma-3 O43741 Q13131 Q9UGI9
Human
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/catalytic subunit alpha-2/subunit beta-1/subunit beta-2/subunit gamma-1/subunit gamma-2/subunit gamma-3 O54950 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078
Mus musculus
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1 P54619 Q13131 Q9Y478
Human
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-2/subunit gamma-1 P54645 P80385 Q9QZH4
Rattus norvegicus
EC50: 3
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-2/subunit gamma-1 O43741 P54619 Q13131
Human
5'-AMP-activated protein kinase catalytic subunit alpha-2/subunit beta-1/subunit gamma-1 P54619 P54646 Q9Y478
Human
5'-AMP-ACTIVATED PROTEIN KINASE SUBUNIT GAMMA-2 O43741 O54950 P54646 Q13131 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078 Q9UGJ0 Q9Y478
EC50: 5
5'-AMP-activated protein kinase catalytic subunit alpha-1/catalytic subunit alpha-2/subunit beta-1/subunit beta-2/subunit gamma-1/subunit gamma-2/subunit gamma-3 O54950 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078
Mus musculus
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-2 Q13131 Q9UGJ0 Q9Y478
Human
EC50: 1
5'-AMP-activated protein kinase catalytic subunit alpha-2/subunit beta-1/subunit gamma-2 P54646 Q9UGJ0 Q9Y478
Human
EC50: 1
5'-AMP-ACTIVATED PROTEIN KINASE SUBUNIT GAMMA-3 O43741 O54950 Q13131 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078 Q9UGI9 Q9Y478
EC50: 3
5'-AMP-activated protein kinase catalytic subunit alpha-1/catalytic subunit alpha-2/subunit beta-1/subunit beta-2/subunit gamma-1/subunit gamma-2/subunit gamma-3 O54950 Q5EG47 Q6PAM0 Q8BGM7 Q8BRK8 Q91WG5 Q9R078
Mus musculus
EC50: 1
Escherichia coli (strain K12)
Neisseria meningitidis
Kd: 8
Klebsiella pneumoniae
Kd: 8
Staphylococcus aureus
Kd: 8
Rattus norvegicus (rat)
Cricetulus griseus (Chinese hamster) (Cricetulus barabensis griseus)
Ki: 53
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
Rattus norvegicus (Rat)
5-HYDROXYTRYPTAMINE RECEPTOR 1B A0A1V4JMG2 A5X5Y0 L8IGV0 O08892 O95264 P08908 P08909 P14842 P19327 P28221 P28222 P28223 P28334 P28335 P28564 P28565 P28566 P30939 P30940 P30994 P31388 P32305 P34969 P35364 P35365 P35563 P41595 P46098 P46636 P47898 P49144 P50406 P79250 P79399 Q13639 Q62758 Q70Z44 Q8WXA8 Q9JJ16 Q9N2B7
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
Rattus norvegicus (Rat)
5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7 P08909 P14842 P19327 P28564 P28565 P30940 P30994 P31388 P32305 P35364 P35365 P35563 Q62758 Q9JJ16
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Cricetulus griseus (Chinese hamster) (Cricetulus barabensis griseus)
Ki: 54
Canis lupus familiaris (Dog) (Canis familiaris)
Ki: 2
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
Rattus norvegicus (Rat)
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
Oryctolagus cuniculus (Rabbit)
IC50: 3
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
Rattus norvegicus (Rat)
5-HYDROXYTRYPTAMINE RECEPTOR 2A A0A1V4J4E5 A5X5Y0 G1SYA7 O46635 O95264 P08908 P08909 P14842 P19327 P28221 P28222 P28223 P28335 P28564 P28565 P28566 P30939 P30940 P30994 P31388 P32305 P34968 P34969 P35363 P35364 P35365 P35563 P41595 P46098 P47898 P49137 P50128 P50129 P50406 Q02152 Q13639 Q14416 Q62758 Q70Z44 Q75Z89 Q8WXA8 Q9JJ16
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7 P08909 P14842 P19327 P28564 P28565 P30940 P30994 P31388 P32305 P35364 P35365 P35563 Q62758 Q9JJ16
Rattus norvegicus (Rat)
Human
Rattus norvegicus (rat)
Human
Mus musculus (Mouse)
Human
IC50: 8
Human
Rattus norvegicus (Rat)
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7 P08909 P14842 P19327 P28564 P28565 P30940 P30994 P31388 P32305 P35364 P35365 P35563 Q62758 Q9JJ16
Rattus norvegicus (Rat)
Human
Mus musculus (Mouse)
Rattus norvegicus (Rat)
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7 P08909 P14842 P19327 P28564 P28565 P30940 P30994 P31388 P32305 P35364 P35365 P35563 Q62758 Q9JJ16
Rattus norvegicus (Rat)
Human
Mus musculus (Mouse)
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7 P08909 P14842 P19327 P28564 P28565 P30940 P30994 P31388 P32305 P35364 P35365 P35563 Q62758 Q9JJ16
Rattus norvegicus (Rat)
Mus musculus (house mouse)
Mus musculus (house mouse)
Human
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7 P08909 P14842 P19327 P28564 P28565 P30940 P30994 P31388 P32305 P35364 P35365 P35563 Q62758 Q9JJ16
Rattus norvegicus (Rat)
Mus musculus (house mouse)
Human
5-HYDROXYTRYPTAMINE RECEPTOR 3C A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
Human
5-HYDROXYTRYPTAMINE RECEPTOR 3D A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-HYDROXYTRYPTAMINE RECEPTOR 3E A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
Human
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7 A5X5Y0 O95264 P08908 P28221 P28222 P28223 P28335 P28566 P30939 P34969 P41595 P46098 P47898 P50406 Q13639 Q70Z44 Q8WXA8
Human
Human
IC50: 3
Curated by BindingDB
Curated by ChEMBL