BDBM217380 CDDO-EA, 3
SMILES CCNC(=O)[C@]12CCC(C)(C)C[C@H]1[C@H]1C(=O)C=C3[C@@]4(C)C=C(C#N)C(=O)C(C)(C)[C@@H]4CC[C@@]3(C)[C@]1(C)CC2
InChI Key InChIKey=RZRQJICXYQPEQJ-YKEYHJQHSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 217380
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human GOAT expressed in baculovirus infected sf9 insect cell membrane using GSSFLC-acrylodan and octanoyl-CoA as substrate preincubated...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair