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Found 2 Enz. Inhib. hit(s) with Target = 'Ghrelin O-acyltransferase' and Ligand = 'BDBM217380'
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM217380(CDDO-EA, 3)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human GOAT expressed in baculovirus infected sf9 insect cell membrane using GSSFLC-acrylodan and octanoyl-CoA as substrate preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM217380(CDDO-EA, 3)
Affinity DataIC50:  8.00E+3nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed