BDBM23738 2-(1-benzyl-5-methoxy-2-methyl-1H-indol-3-yl)acetamide::CHEMBL346855::Indole Derivative, 1
SMILES COc1ccc2n(Cc3ccccc3)c(C)c(CC(N)=O)c2c1
InChI Key InChIKey=RUPYVFAPAMOERU-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 23738
Affinity DataIC50: 540nMpH: 8.0 T: 2°CAssay Description:Phospholipase A2 was assayed using unlabeled lipids as substrate and 1-anilinonaphthalene-8-sulfonate (ANS) as a probe for the interfacial reaction. ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:Inhibition of Human Nonpancreatic Secretory Phospholipase A2 through Chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human LTA4H aminopeptidase activity using Ala-p-nitroanilide as substrate incubated for 2 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Inhibition of human nonpancreatic secretory phospholipase A2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine as substrate after 10 mins by spectrop...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human LTA4H epoxide hydrolase activity using LTA4 as substrate incubated for 15 mins prior to substrate addition measured after 10 mins...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair