BDBM285025 2-methyl-4-pyridin-2-ylisoquinolin-1-one::US10023592, Example 70::US10941160, Example 70

SMILES Cn1cc(-c2ccccn2)c2ccccc2c1=O


Data  3 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 285025   

TargetBromodomain-containing protein 4(Homo sapiens (Human))
Celgene Quanticel Research

Curated by ChEMBL
LigandPNGBDBM285025(2-methyl-4-pyridin-2-ylisoquinolin-1-one | US10023...)
Show SMILES Cn1cc(-c2ccccn2)c2ccccc2c1=O
Show InChI InChI=1S/C15H12N2O/c1-17-10-13(14-8-4-5-9-16-14)11-6-2-3-7-12(11)15(17)18/h2-10H,1H3
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of His-tagged human BRD4-BD1 using H4K5acK8acK12acK16ac as substrate preincubated for 30 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid