BDBM293449 US10106527, Compound 52::US10544128, Compound 52::US11548872, Compound 52::US20230286945, Compound 52::US9951048, Compound 52

SMILES CC(C)Oc1ccc(cc1)C(=O)Nc1cc2cc(ccc2cn1)-c1cnc2CNCCn12

InChI Key InChIKey=XLPAJQNQDWMMLT-UHFFFAOYSA-N

Data  10 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 293449   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Biosplice Therapeutics

US Patent
LigandPNGBDBM293449(US10106527, Compound 52 | US10544128, Compound 52 ...)
Affinity DataEC50:  3.10nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies?a Divis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent