BDBM293449 US10106527, Compound 52::US10544128, Compound 52::US11548872, Compound 52::US20230286945, Compound 52::US9951048, Compound 52
SMILES CC(C)Oc1ccc(cc1)C(=O)Nc1cc2cc(ccc2cn1)-c1cnc2CNCCn12
InChI Key InChIKey=XLPAJQNQDWMMLT-UHFFFAOYSA-N
Data 10 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 293449
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed
US Patent
Samumed
US Patent
Affinity DataEC50: 3.10nMT: 2°CAssay Description:Briefly, recombinant DYRK1A kinase, ATP and Ser/Thr peptide 18 were prepared in 1× Kinase buffer to final concentrations of 0.19 μg/mL, 30 μ...More data for this Ligand-Target Pair
Affinity DataEC50: 4.32E+3nMT: 2°CAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 ...More data for this Ligand-Target Pair