BDBM393487 US9963460, 13

SMILES CN(Cc1ccccc1)C(=O)C1=C[C@]23CC[C@]1(O)[C@@H]1Oc4c5c(C[C@H]2N(CC2CC2)CC[C@@]315)ccc4O

InChI Key InChIKey=KZYGDXSSQSUQMI-RZBRXQIYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 393487   

TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

US Patent
LigandPNGBDBM393487(US9963460, 13)
Affinity DataEC50:  0.00280nMAssay Description:In a [3SS] GTPγS binding test, the opioid receptor agonist activity of test compounds based on a GTP-GDP exchange reaction was evaluated. In the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

US Patent
LigandPNGBDBM393487(US9963460, 13)
Affinity DataEC50:  1.70nMAssay Description:In a [3SS] GTPγS binding test, the opioid receptor agonist activity of test compounds based on a GTP-GDP exchange reaction was evaluated. In the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

US Patent
LigandPNGBDBM393487(US9963460, 13)
Affinity DataEC50:  2.77nMAssay Description:In a [3SS] GTPγS binding test, the opioid receptor agonist activity of test compounds based on a GTP-GDP exchange reaction was evaluated. In the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent