BDBM50198757 CHEMBL363142
SMILES [#6]-c1cc(-[#8])cc(-[#6])c1-[#6]-[#6](-[#7])-[#6](=O)-[#7]-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6](-[#7])=O
InChI Key InChIKey=FIAKHZXVLBNZLW-ZAEYVGPMSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50198757
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.143nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]U69,593 from KOR in guinea pig brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Displacement of [3H]DSLET from DOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at MOR in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair