TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.143nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at MOR in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionsMore data for this Ligand-Target Pair